SCHEMBL7016571

SCHEMBL7016571

Cn1c(SCc2ccc(C(=O)c3ccc(Cl)cc3)cc2)nc2c(ccn2C)c1=O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 2/20 0.54
MAOB P27338 2/20 0.54
RXFP1 Q9HBX9 1/20 0.48
ALDH1A1 P00352 6/20 0.45
MAPT P10636 5/20 0.45
HTT P42858 2/20 0.45
NPSR1 Q6W5P4 2/20 0.45
LMNA P02545 3/20 0.45
TP53 P04637 2/20 0.45
THRB P10828 1/20 0.45
MEN1 O00255 5/20 0.44
KMT2A Q03164 5/20 0.44
RAB9A P51151 2/20 0.43
ALDH1A2 O94788 1/20 0.43
ALDH1A3 P47895 1/20 0.43
TSHR P16473 5/20 0.43
HSD17B10 Q99714 5/20 0.43
KDM1A O60341 1/20 0.43
HDAC3 O15379 1/20 0.42
HDAC4 P56524 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7012122 0.89 MAOA (0.54) MAOAMAOBRXFP1ALDH1A1MAPT
SCHEMBL7011645 0.84 ALDH1A1 (0.58) MAOAMAOBRXFP1ALDH1A1MAPT
SCHEMBL7011866 0.83 MAOA (0.46) MAOAMAOBRXFP1ALDH1A1MAPT
SCHEMBL7013210 0.82 MEN1 (0.53) MAOAMAOBMAPTNPSR1LMNA
SCHEMBL7015339 0.82 KMT2A (0.68) MAPTNPSR1LMNATP53MEN1
SCHEMBL7011263 0.81 MAOA (0.52) MAOAMAOBRXFP1ALDH1A1MAPT
SCHEMBL9060596 0.80 MAOA (0.52) MAOAMAOBRXFP1ALDH1A1MAPT
SCHEMBL7013087 0.80 ALDH1A1 (0.36) ALDH1A1MAPTHTTNPSR1LMNA
SCHEMBL7011002 0.80 MEN1 (0.48) MAOAMAOBRXFP1ALDH1A1MAPT
SCHEMBL7009666 0.80 MAOA (0.47) MAOAMAOBRXFP1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed