SCHEMBL7019246

SCHEMBL7019246

Cc1cccc2c1[N]CCCC2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.41
TSHR P16473 2/20 0.39
BCL2L1 Q07817 1/20 0.38
BAD Q92934 1/20 0.38
ALOX12 P18054 1/20 0.37
ALDH1A1 P00352 4/20 0.36
LMNA P02545 4/20 0.36
HPGD P15428 2/20 0.36
KDM4E B2RXH2 1/20 0.36
NR4A1 P22736 1/20 0.36
HTT P42858 1/20 0.36
CCNA2 P20248 1/20 0.36
CDK2 P24941 1/20 0.36
CDK5 Q00535 1/20 0.36
CDK5R1 Q15078 1/20 0.36
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
CYP1A2 P05177 1/20 0.34
CYP2A6 P11509 1/20 0.34
USP2 O75604 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1091403 0.94 ALOX12 (0.38) POLBTSHRBCL2L1BADALOX12
SCHEMBL1936960 0.86 CYP1A2 (0.44) POLBTSHRALOX12ALDH1A1LMNA
SCHEMBL5544284 0.71 NOS3 (0.39) TSHRBCL2L1BAD
SCHEMBL5545432 0.71 TSHR (0.36) TSHRBCL2L1BADMEN1KMT2A
SCHEMBL5539619 0.71 NOS3 (0.37) TSHRBCL2L1BAD
SCHEMBL12043594 0.71 CYP2A6 (0.36) POLBALOX12ALDH1A1LMNAHPGD
SCHEMBL249643 0.71 BCL2L1 (0.48) TSHRBCL2L1BADALDH1A1LMNA
SCHEMBL8860490 0.71 NOS3 (0.43) POLBTSHRBCL2L1BADALDH1A1
SCHEMBL5545601 0.71 ACHE (0.41) POLBTSHRBCL2L1BADCYP1A2
SCHEMBL301029 0.70 NPC1 (0.41) KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1051415-B1 BENZAMIDE DERIVATIVES AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO (JP) 2003-09-24 EP disclosed
US-6495542-B1 SUCH AS 2-METHOXY-N-(2-METHYL-1H-BENZIMIDAZOL-4-YL)-4-(2,3,4,5-TETRAHYDRO-5-OXO-1H-1-BENZAZEPIN-1-YL)CARBONYL-BENZAM IDE; HYPERTENSION, HEART FAILURE, RENAL INSUFFICIENCY, EDEMA, ASCITES, VASOPRESSIN PARASECRETION SYNDROME FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-12-17 US disclosed