SCHEMBL8860490

SCHEMBL8860490

Nc1cccc2c1[N]CCC2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 3/20 0.43
KDM4E B2RXH2 5/20 0.42
ALDH1A1 P00352 5/20 0.42
HPGD P15428 4/20 0.42
MAPT P10636 3/20 0.42
KMT2A Q03164 3/20 0.42
LMNA P02545 2/20 0.42
GAA P10253 2/20 0.42
MEN1 O00255 2/20 0.42
HSD17B10 Q99714 4/20 0.38
HIF1A Q16665 1/20 0.38
TSHR P16473 4/20 0.36
CYP3A4 P08684 3/20 0.36
TDP1 Q9NUW8 2/20 0.36
CD44 P16070 1/20 0.35
NOS2 P35228 2/20 0.33
POLB P06746 2/20 0.32
NPC1 O15118 1/20 0.32
GLA P06280 1/20 0.32
PTBP1 P26599 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL249643 0.76 BCL2L1 (0.48) NOS3ALDH1A1HPGDMAPTKMT2A
SCHEMBL5545432 0.76 TSHR (0.36) NOS3KMT2AMEN1TSHRBCL2L1
SCHEMBL5544284 0.76 NOS3 (0.39) NOS3TSHRTDP2BCL2L1BAD
SCHEMBL5545601 0.76 ACHE (0.41) NOS3TSHRPOLBNPSR1BCL2L1
SCHEMBL5539619 0.76 NOS3 (0.37) NOS3TSHRNOS2BCL2L1BAD
SCHEMBL1091403 0.76 ALOX12 (0.38) NOS3KDM4EALDH1A1HPGDMAPT
Bromide SCHEMBL11832552 0.74 BCL2L1 (0.47) NOS3ALDH1A1HPGDMAPTKMT2A
SCHEMBL301029 0.72 NPC1 (0.41) KDM4ENPC1
SCHEMBL7019246 0.71 POLB (0.41) KDM4EALDH1A1HPGDMAPTKMT2A
SCHEMBL1525254 0.71 ALDH1A1 (0.47) KDM4EALDH1A1MAPTKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5668131-A CONTROLLING HELICOBACTER BACTERIA BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1997-09-16 US disclosed
EP-0731801-A1 SUBSTITUTED AMINOALKYLAMINOPYRIDINES Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1996-09-18 EP disclosed
WO-1996000224-A1 4-S- AND N-SUBSTITUTED 6-ALKYLPYRIDINES FOR CONTROLLING HELICOBACTER BACTERIA BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1996-01-04 WO disclosed
WO-1995015324-A1 SUBSTITUTED AMINOALKYLAMINOPYRIDINES BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1995-06-08 WO disclosed