SCHEMBL702242

SCHEMBL702242

COC(=O)c1ccc(OC(=O)c2ccc(O)cc2)cc1

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 4/20 0.77
CA2 P00918 4/20 0.77
CA12 O43570 1/20 0.77
CA7 P43166 1/20 0.77
CA9 Q16790 1/20 0.77
CA14 Q9ULX7 1/20 0.77
ACR P10323 3/20 0.61
HGFAC Q04756 1/20 0.61
PRSS1 P07477 1/20 0.59
KMT2A Q03164 4/20 0.58
ALDH1A1 P00352 2/20 0.57
LMNA P02545 2/20 0.57
GAA P10253 1/20 0.57
L3MBTL1 Q9Y468 1/20 0.57
MAPT P10636 2/20 0.56
KDM4E B2RXH2 1/20 0.55
POLB P06746 1/20 0.55
TDP1 Q9NUW8 1/20 0.53
STS P08842 1/20 0.51
ELANE P08246 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10834543 1.00 CA1 (0.77) CA1CA2CA12CA7CA9
SCHEMBL16426422 1.00 CA1 (0.77) CA1CA2CA12CA7CA9
SCHEMBL28480069 0.98 CA1 (0.74) CA1CA2CA12CA7CA9
SCHEMBL15214832 0.95 CA1 (0.69) CA1CA2CA12CA7CA9
SCHEMBL7518320 0.92 CA1 (0.72) CA1CA2CA12CA7CA9
SCHEMBL16078330 0.90 MAPT (0.75) CA1CA2CA12CA7CA9
SCHEMBL9696072 0.90 HSD17B10 (0.59) CA1CA2CA12CA7CA9
SCHEMBL688276 0.90 HSD17B10 (0.59) CA1CA2CA12CA7CA9
SCHEMBL16493489 0.90 HSD17B10 (0.59) CA1CA2CA12CA7CA9
SCHEMBL740606 0.90 HSD17B10 (0.59) CA1CA2CA12CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 32 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3621958-B1 PHOTOCHROMIC INDENO FUSED PHENANTHRENOPYRAN COMPOUNDS TRANSITIONS OPTICAL LTD (IE) 2024-07-10 EP disclosed
EP-3268375-B1 PHOTOCHROMIC THIENOCHROMENE COMPOUNDS TRANSITIONS OPTICAL INC (US) 2022-06-15 EP disclosed
EP-3071576-B9 PHOTOCHROMIC INDENO-FUSED RING PYRAN COMPOUNDS TRANSITIONS OPTICAL INC (US) 2021-12-22 EP disclosed
EP-3071576-B1 PHOTOCHROMIC INDENO-FUSED RING PYRAN COMPOUNDS TRANSITIONS OPTICAL INC (US) 2021-08-18 EP disclosed
US-20200048216-A1 Photochromic Indeno Fused Phenanthrenopyran Compounds TRANSITIONS OPTICAL, LTD. (IE) 2020-02-13 US disclosed
EP-3071550-B1 METHOD OF PREPARING FUSED RING INDENO COMPOUNDS TRANSITIONS OPTICAL INC (US) 2019-03-13 EP disclosed
US-20180051037-A1 Photochromic Thienochromene Compounds TRANSITIONS OPTICAL, INC. 2018-02-22 US disclosed
US-9630902-B2 Method of preparing fused ring indeno compounds TRANSITIONS OPTICAL, INC. (US) 2017-04-25 US disclosed
US-20160209561-A1 Photochromic Articles That Include Photochromic-Dichroic Materials TRANSITIONS OPTICAL, INC. 2016-07-21 US disclosed
US-9334439-B2 Photochromic articles that include photochromic-dichroic materials TRANSITIONS OPTICAL, INC. (US) 2016-05-10 US disclosed
US-8575097-B2 Exendin variant and conjugate thereof PEGBIO CO., LTD. (CN) 2013-11-05 US disclosed
US-8455061-B2 Optically active compound having polymerizable group and its polymer JNC CORPORATION (JP) 2013-06-04 US disclosed
US-20120196795-A1 NOVEL EXENDIN VARIANT AND CONJUGATE THEREOF PEGBIO CO., LTD. (CN) 2012-08-02 US disclosed
EP-2423223-A1 NOVEL EXENDIN VARIANT AND CONJUGATE THEREOF Pegbio Co., Ltd. (CN) 2012-02-29 EP disclosed
EP-1613317-A1 COMBINATION OF A MACROLIDE AND A LOCAL ANESTHETIC FOR THE TREATMENT OF DERMATOLOGICAL DISEASES Novartis AG (CH) 2006-01-11 EP disclosed
WO-2004087144-A1 COMBINATION OF A MACROLIDE AND A LOCAL ANESTHETIC FOR THE TREATMENT OF DERMATOLOGICAL DISEASES NOVARTIS AG (CH) 2004-10-14 WO disclosed
EP-0352293-A4 NON-CRYSTALLINE MINOXIDIL COMPOSITION AND METHOD OF APPLICATION 1991-03-20 EP disclosed
EP-0352293-A1 NON-CRYSTALLINE MINOXIDIL COMPOSITION AND METHOD OF APPLICATION LIPOSOME TECHNOLOGY, INC. (US) 1990-01-31 EP disclosed
US-4828837-A Non-crystalline minoxidil composition, its production and application LIPOSOME TECHNOLOGY, INC. (US) 1989-05-09 US disclosed
WO-1988007362-A1 NON-CRYSTALLINE MINOXIDIL COMPOSITION AND METHOD OF APPLICATION LIPOSOME TECHNOLOGY, INC. (US) 1988-10-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200048216-A1 Photochromic Indeno Fused Phenanthrenopyran Compounds ALDH1A2, RB1, INCENP CA1 3567/4885CA2 1663/4885CA12 2526/4885
US-20120196795-A1 NOVEL EXENDIN VARIANT AND CONJUGATE THEREOF GLP1R, IAPP, GIPR CA1 4704/4885CA2 4112/4885CA12 1780/4885
US-20180051037-A1 Photochromic Thienochromene Compounds CRY1, CRY2, TERT CA1 4264/4885CA2 3806/4885CA12 4355/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.