SCHEMBL7023007

SCHEMBL7023007

NC(=O)NS(=O)(=O)c1ccccc1-c1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 2/20 0.54
BCAT2 O15382 1/20 0.46
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
EDNRA P25101 5/20 0.43
EDNRB P24530 4/20 0.43
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
MMP1 P03956 1/20 0.42
MMP2 P08253 1/20 0.42
MMP9 P14780 1/20 0.42
MMP8 P22894 1/20 0.42
MMP13 P45452 1/20 0.42
BCL2 P10415 1/20 0.41
BCL2L1 Q07817 1/20 0.41
MCL1 Q07820 1/20 0.41
BCL2A1 Q16548 1/20 0.41
BCL2L2 Q92843 1/20 0.41
UCHL1 P09936 1/20 0.40
USP30 Q70CQ3 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8240985 0.86 CASP1 (0.56) CASP1BCAT2MEN1KMT2AEDNRA
SCHEMBL9682375 0.85 CASP1 (0.49) CASP1BCAT2EDNRAEDNRBBCL2
SCHEMBL5147607 0.83 CASP1 (0.54) CASP1EDNRAEDNRBCA1CA2
SCHEMBL10729804 0.80 CA1 (0.55) MEN1KMT2ACA1CA2MMP1
SCHEMBL10916572 0.80 CASP1 (0.51) CASP1EDNRAEDNRBFGFR1SRC
SCHEMBL10915661 0.80 CASP1 (0.45) CASP1BCAT2MEN1KMT2AEDNRA
SCHEMBL29537027 0.80 CA2 (0.58) CASP1EDNRAEDNRBCA1CA2
SCHEMBL1767981 0.80 CA2 (0.58) CASP1EDNRAEDNRBCA1CA2
SCHEMBL8997291 0.79 CASP1 (0.50) CASP1EDNRAEDNRBCA1CA2
SCHEMBL418847 0.78 CASP1 (0.51) CASP1EDNRAEDNRBCA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 23 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4586951-A PLANT GROWTH REGULATORS FOR RICE FIELDS NIHON TOKUSHU NOYAKU SEIZO K.K. (JP) 1986-05-06 US claimed
EP-0560177-B1 Imidazole derivatives having biphenylsulphonylurea or biphenylsulfonylurethane side chains, process for their production and use thereof HOECHST AG (DE) 2003-01-08 EP disclosed
EP-1183236-A1 CINNAMOYLAMINOALKYL-SUBSTITUTED BENZENESULFONAMIDE DERIVATIVES Aventis Pharma Deutschland GmbH (DE) 2002-03-06 EP disclosed
US-6350778-B1 CARDIOVASCULAR DISORDERS AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2002-02-26 US disclosed
WO-2000071513-A1 CINNAMOYLAMINOALKYL-SUBSTITUTED BENZENESULFONAMIDE DERIVATIVES AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2000-11-30 WO disclosed
US-5604251-A Imidazole derivatives with a biphenylsulfonylurea or biphenylsulfonylurethane side chain and their use as angitensin II receptors HOECHST AKTIENGESELLSCHAFT (DE) 1997-02-18 US disclosed
US-5604251-A Imidazole derivatives with a biphenylsulfonylurea or biphenylsulfonylurethane side chain and their use as angitensin II receptors HOECHST AKTIENGESELLSCHAFT (DE) 1997-02-18 US disclosed
US-5604251-A Imidazole derivatives with a biphenylsulfonylurea or biphenylsulfonylurethane side chain and their use as angitensin II receptors HOECHST AKTIENGESELLSCHAFT (DE) 1997-02-18 US disclosed
EP-0560177-A1 Imidazole derivatives having biphenylsulphonylurea or biphenylsulfonylurethane side chains, process for their production and use thereof HOECHST AKTIENGESELLSCHAFT (DE) 1993-09-15 EP disclosed
US-4810282-A 3-ORTHO-(ISOXAZOLYL,ISOTHIAZOLYL, PYRAZOLYL,THIADIAZOLYL, OXADIAZOLYL AND TRIAZOLYL BENZENESULFONUREYLENE-1,2,4-TRIAZOLES E. I. DU PONT DE NEMOURS AND COMPANY (US) 1989-03-07 US disclosed
US-4695311-A Herbicidal sulfonamides E. I. DU PONT DE NEMOURS AND COMPANY (US) 1987-09-22 US disclosed
US-4606755-A Herbicidal sulfonamides E. I. DU PONT DE NEMOURS AND COMPANY (US) 1986-08-19 US disclosed
US-4600792-A PHENYL 2-BIPHENYLYLSULFONYLCARBAMATE, HERBICIDES NIHON TOKUSHU NOYAKU SEIZO K.K. (JP) 1986-07-15 US disclosed
US-4600792-A PHENYL 2-BIPHENYLYLSULFONYLCARBAMATE, HERBICIDES NIHON TOKUSHU NOYAKU SEIZO K.K. (JP) 1986-07-15 US disclosed
US-4592775-A Containing hetero ring substitution E. I. DU PONT DE NEMOURS AND COMPANY (US) 1986-06-03 US disclosed
EP-0158248-A3 PROCESS FOR THE PREPARATION OF BIPHENYLSULFONYL UREA DERIVATIVES, THEIR INTERMEDIATES AND PROCESS FOR THE PREPARATION OF THE INTERMEDIATES NIHON TOKUSHU NOYAKU SEIZO K.K. (JP) 1986-02-12 EP disclosed
EP-0158248-A2 Process for the preparation of biphenylsulfonyl urea derivatives, their intermediates and process for the preparation of the intermediates NIHON TOKUSHU NOYAKU SEIZO K.K. (JP) 1985-10-16 EP disclosed
US-4511392-A N--/PYRIMIDIN-2-YLAMINOCARBENYL/-HETERO-SUBSTITUETED BENZENSESULFO E. I. DU PONT DE NEMOURS AND COMPANY (US) 1985-04-16 US disclosed
US-4460401-A PLANT GROWTH REGULATORS E. I. DU PONT DE NEMOURS AND COMPANY (US) 1984-07-17 US disclosed
EP-0083975-A2 Herbicidal sulfonamides E.I. DU PONT DE NEMOURS AND COMPANY (US) 1983-07-20 EP disclosed