SCHEMBL7027296

SCHEMBL7027296

COc1ccccc1N1CCN(C(Cc2ccccc2)C(N)=O)CC1

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.56
ADRA1D P25100 1/20 0.52
ADRA1A P35348 1/20 0.52
ADRA1B P35368 1/20 0.52
ALDH1A1 P00352 4/20 0.52
TSHR P16473 1/20 0.52
LMNA P02545 1/20 0.52
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51
HTR1A P08908 1/20 0.50
KDM4E B2RXH2 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
HTR7 P34969 1/20 0.50
RAB9A P51151 1/20 0.49
DRD2 P14416 1/20 0.49
DRD4 P21917 1/20 0.49
DRD3 P35462 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28201210 0.86 TSHR (0.58) POLBADRA1DADRA1AADRA1BALDH1A1
SCHEMBL9331896 0.86 PKM (0.58) POLBADRA1DADRA1AADRA1BALDH1A1
SCHEMBL8443576 0.81 ADRA1D (0.56) POLBADRA1DADRA1AADRA1BALDH1A1
SCHEMBL6936789 0.80 ALDH1A1 (0.58) POLBALDH1A1TSHRLMNAMEN1
Hydrochloric Acid SCHEMBL7029028 0.78 POLB (0.55) POLBADRA1DADRA1AADRA1BALDH1A1
Hydrochloric Acid SCHEMBL6706983 0.78 ALDH1A1 (0.63) POLBALDH1A1TSHRLMNAMEN1
Hydrochloric Acid SCHEMBL6706985 0.78 ALDH1A1 (0.63) POLBALDH1A1TSHRLMNAMEN1
SCHEMBL11509122 0.78 GAA (0.61) POLBADRA1DADRA1AADRA1BALDH1A1
SCHEMBL8492185 0.77 DRD2 (0.52) POLBALDH1A1TSHRLMNAMEN1
Hydrochloric Acid SCHEMBL11817434 0.77 GAA (0.60) POLBADRA1DADRA1AADRA1BALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1276731-A2 BRANCHED ADAMANTYL AND NORADAMANTYL ARYL- AND ARALKYLPIPERAZINES WITH SEROTONIN 5-HT 1A ACTIVITY Wyeth (US) 2003-01-22 EP claimed
WO-2001034586-A2 BRANCHED ADAMANTYL AND NORADAMANTYL ARYL- AND ARALKYLPIPERAZINES WITH SEROTONIN 5-HT1A ACTIVITY WYETH (US) 2001-05-17 WO claimed