SCHEMBL7039451

SCHEMBL7039451

C=CCn1c(=O)c2c(nc(-c3ccccc3)n2CC=C)n(C)c1=O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 5/20 0.86
ALDH1A1 P00352 2/20 0.86
KDM4E B2RXH2 1/20 0.62
MAPT P10636 1/20 0.62
THRB P10828 1/20 0.62
HPGD P15428 1/20 0.62
BLM P54132 1/20 0.62
HSD17B10 Q99714 1/20 0.62
RCE1 Q9Y256 1/20 0.62
SMN1; SMN2 Q16637 2/20 0.57
CYP1A2 P05177 1/20 0.57
CYP3A4 P08684 1/20 0.57
CYP2C9 P11712 1/20 0.57
CYP2C19 P33261 1/20 0.57
POLB P06746 1/20 0.57
ADORA2A P29274 2/20 0.54
PKM P14618 2/20 0.54
LMNA P02545 1/20 0.53
MAPK1 P28482 1/20 0.53
HTT P42858 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5411870 0.93 ADORA2B (1.00) ADORA2BALDH1A1KDM4EMAPTTHRB
SCHEMBL7037071 0.88 ADORA2B (0.67) ADORA2BALDH1A1KDM4EMAPTTHRB
SCHEMBL7034529 0.78 ADORA2B (0.55) ADORA2BALDH1A1KDM4EMAPTTHRB
SCHEMBL1319913 0.77 ALDH1A1 (1.00) ADORA2BALDH1A1KDM4EMAPTTHRB
SCHEMBL7034258 0.76 ADORA2B (0.56) ADORA2BALDH1A1KDM4EMAPTTHRB
SCHEMBL9765909 0.76 ADORA2B (1.00) ADORA2BALDH1A1KDM4EHPGDBLM
SCHEMBL7030152 0.75 ADORA2B (0.70) ADORA2BALDH1A1HPGDSMN1; SMN2ADORA2A
SCHEMBL19666778 0.75 ALDH1A1 (0.68) ADORA2BALDH1A1KDM4EMAPTTHRB
SCHEMBL7034532 0.74 POLB (0.58) ADORA2BALDH1A1MAPTHSD17B10SMN1; SMN2
SCHEMBL17626266 0.73 ADORA2B (0.67) ADORA2BALDH1A1HPGDSMN1; SMN2ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0956855-B1 Immunosuppressive effects of 8 substituted xanthine derivatives LEUVEN K U RES & DEV (BE) 2003-03-12 EP claimed