SCHEMBL7041774

SCHEMBL7041774

CCC1CCCCN1CCn1c(N2CCCNCC2)nc2c(OC(N)=O)cccc21

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.37
THRB P10828 1/20 0.35
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
NPC1 O15118 1/20 0.34
TERT O14746 2/20 0.34
HTR3A P46098 1/20 0.33
PARP1 P09874 1/20 0.33
TP53 P04637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7040063 0.98 SMN1; SMN2 (0.36) SMN1; SMN2THRBCYP1A2CYP3A4CYP2D6
SCHEMBL7706399 0.88 PARP1 (0.43) THRBNPC1PARP1
SCHEMBL7041918 0.87 PARP1 (0.40) SMN1; SMN2THRBTERTPARP1TP53
SCHEMBL7046250 0.87 PARP1 (0.38) SMN1; SMN2THRBNPC1TERTPARP1
SCHEMBL7708432 0.85 PARP1 (0.45) THRBTERTPARP1
SCHEMBL7046777 0.85 HTR3A (0.39) HTR3A
SCHEMBL7041579 0.85 JAK2 (0.40) SMN1; SMN2THRBCYP1A2CYP3A4CYP2D6
SCHEMBL7037841 0.84 HTR3A (0.38) HTR3APARP1
SCHEMBL7042010 0.84 FLT3 (0.41) CYP1A2CYP3A4HTR3A
SCHEMBL7036855 0.83 HTR3A (0.40) HTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133477-B1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS ABBOTT GMBH & CO KG (DE) 2004-02-18 EP disclosed
EP-1133477-A1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2001-09-19 EP disclosed
WO-2000032579-A1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2000-06-08 WO disclosed