SCHEMBL7042010

SCHEMBL7042010

CCn1c(N2CCCNCC2)nc2c(OC(N)=O)cccc21

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
FLT3 P36888 1/20 0.41
KCNH2 Q12809 1/20 0.41
PIM1 P11309 1/20 0.40
SOS1 Q07889 1/20 0.37
HTR3A P46098 6/20 0.37
CHRNB2 P17787 1/20 0.36
CHRNA4 P43681 1/20 0.36
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C19 P33261 1/20 0.36
IKBKB O14920 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7045272 0.96 FLT3 (0.44) FLT3KCNH2PIM1SOS1HTR3A
SCHEMBL7036855 0.89 HTR3A (0.40) PIM1SOS1HTR3ACHRNB2CHRNA4
SCHEMBL7044695 0.89 HTR3A (0.40) PIM1SOS1HTR3ACHRNB2CHRNA4
SCHEMBL7045753 0.89 HTR3A (0.38) SOS1HTR3ACHRNB2CHRNA4KMT2A
SCHEMBL7043340 0.88 CHRNB2 (0.39) HTR3ACHRNB2CHRNA4KMT2AMEN1
SCHEMBL7046777 0.87 HTR3A (0.39) HTR3ACHRNB2CHRNA4
SCHEMBL7037841 0.87 HTR3A (0.38) HTR3AKMT2AMEN1
SCHEMBL7042935 0.85 HTR3A (0.42) KCNH2PIM1SOS1HTR3A
SCHEMBL5621918 0.85 PARP1 (0.44) FLT3KCNH2PIM1CHRNB2CHRNA4
SCHEMBL7042964 0.85 HTR3A (0.42) KCNH2PIM1SOS1HTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133477-B1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS ABBOTT GMBH & CO KG (DE) 2004-02-18 EP disclosed