SCHEMBL7108289

SCHEMBL7108289

N#Cc1ccc(-c2cnc3cccc(C(N)=O)c3n2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 12/20 1.00
PARP2 Q9UGN5 1/20 1.00
CASP1 P29466 1/20 0.48
ATR Q13535 2/20 0.46
CSF1R P07333 2/20 0.46
MYC P01106 1/20 0.43
JAK2 O60674 1/20 0.42
SCN9A Q15858 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7112515 0.85 PARP1 (1.00) PARP1PARP2
SCHEMBL7111338 0.85 PARP1 (0.80) PARP1PARP2
SCHEMBL7042977 0.84 PARP1 (0.78) PARP1PARP2CASP1CSF1R
SCHEMBL424209 0.84 PARP1 (0.81) PARP1PARP2CASP1ATR
SCHEMBL7045309 0.84 PARP1 (0.78) PARP1PARP2ATRCSF1R
SCHEMBL31602072 0.84 PARP1 (0.81) PARP1PARP2CASP1ATR
SCHEMBL7107333 0.81 PARP1 (1.00) PARP1PARP2CASP1CSF1R
SCHEMBL7045177 0.81 PARP1 (1.00) PARP1PARP2CASP1ATRCSF1R
SCHEMBL7043497 0.80 PARP1 (0.71) PARP1PARP2ATR
SCHEMBL7042013 0.80 PARP1 (0.71) PARP1PARP2CASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003007959-A1 QUINOXALINE DERIVATIVES WHICH HAVE PARP INHIBITORY ACTION FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-01-30 WO disclosed