SCHEMBL7045309

SCHEMBL7045309

NC(=O)c1cccc2ncc(-c3ccc(F)cc3)nc12

nearest known ligand 0.78

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 13/20 0.78
PARP2 Q9UGN5 2/20 0.73
NOS1 P29475 1/20 0.43
ATR Q13535 1/20 0.43
CSF1R P07333 1/20 0.42
DHODH Q02127 1/20 0.42
MAP4K4 O95819 1/20 0.41
GRM2 Q14416 1/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
MAPK1 P28482 1/20 0.41
HSD17B10 Q99714 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
AURKA O14965 1/20 0.41
RPS6KB1 P23443 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7112515 0.88 PARP1 (1.00) PARP1PARP2DHODH
SCHEMBL7111338 0.87 PARP1 (0.80) PARP1PARP2DHODHALDH1A1
SCHEMBL7042977 0.86 PARP1 (0.78) PARP1PARP2CSF1RDHODHGRM2
SCHEMBL424209 0.86 PARP1 (0.81) PARP1PARP2ATRDHODHMAP4K4
SCHEMBL31602072 0.86 PARP1 (0.81) PARP1PARP2ATRDHODHMAP4K4
SCHEMBL7107333 0.86 PARP1 (1.00) PARP1PARP2CSF1RAURKARPS6KB1
SCHEMBL7108289 0.84 PARP1 (1.00) PARP1PARP2ATRCSF1R
SCHEMBL7045177 0.83 PARP1 (1.00) PARP1PARP2ATRCSF1RALDH1A1
SCHEMBL7043497 0.82 PARP1 (0.71) PARP1PARP2ATRDHODHMAPK1
SCHEMBL7042013 0.82 PARP1 (0.71) PARP1PARP2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003007959-A1 QUINOXALINE DERIVATIVES WHICH HAVE PARP INHIBITORY ACTION FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-01-30 WO disclosed