SCHEMBL7044209

SCHEMBL7044209

COc1ccc(-c2c(-c3ccccc3Cl)nc(-c3ccccc3Cl)n2-n2c(-c3ccccc3Cl)nc(-c3ccccc3Cl)c2-c2ccc(OC)c(OC)c2)cc1OC

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.54
ALDH1A1 P00352 4/20 0.54
RAB9A P51151 4/20 0.54
L3MBTL1 Q9Y468 3/20 0.54
MEN1 O00255 3/20 0.54
KMT2A Q03164 3/20 0.54
TP53 P04637 3/20 0.54
SMN1; SMN2 Q16637 3/20 0.54
TSHR P16473 2/20 0.54
PDE4A P27815 1/20 0.49
PIK3CD O00329 1/20 0.43
MAPT P10636 1/20 0.43
PDE10A Q9Y233 2/20 0.43
ACACA Q13085 1/20 0.42
KDM4E B2RXH2 3/20 0.42
HPGD P15428 2/20 0.42
HSD17B10 Q99714 2/20 0.42
MAPK1 P28482 1/20 0.42
NPSR1 Q6W5P4 1/20 0.41
PDE2A O00408 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29373643 0.94 L3MBTL1 (0.50) NPC1ALDH1A1RAB9AL3MBTL1MEN1
SCHEMBL62627 0.94 L3MBTL1 (0.50) NPC1ALDH1A1RAB9AL3MBTL1MEN1
SCHEMBL28767208 0.90 ALDH1A1 (0.54) NPC1ALDH1A1RAB9AL3MBTL1MEN1
SCHEMBL7897274 0.87 L3MBTL1 (0.53) NPC1ALDH1A1RAB9AL3MBTL1MEN1
SCHEMBL29732925 0.87 L3MBTL1 (0.53) NPC1ALDH1A1RAB9AL3MBTL1MEN1
SCHEMBL16365751 0.79 L3MBTL1 (0.43) NPC1ALDH1A1RAB9AL3MBTL1MEN1
SCHEMBL29895740 0.79 L3MBTL1 (0.43) NPC1ALDH1A1RAB9AL3MBTL1MEN1
SCHEMBL3083486 0.78 L3MBTL1 (0.45) NPC1ALDH1A1RAB9AL3MBTL1MEN1
SCHEMBL31734215 0.78 L3MBTL1 (0.43) NPC1ALDH1A1RAB9AL3MBTL1MEN1
SCHEMBL16355181 0.78 L3MBTL1 (0.43) NPC1ALDH1A1RAB9AL3MBTL1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2976372-B1 ADHESIVE COMPOSITION BASED ON A POLYESTER URETHANE, AND POLYESTER URETHANE FRAUNHOFER GES FORSCHUNG (DE) 2020-06-03 EP claimed
EP-1000959-B1 Polyetherquat functional polysiloxanes GOLDSCHMIDT AG TH (DE) 2003-04-16 EP claimed
US-6180319-B1 APPLYING AQUEOUS-DEVELOPABLE PHOTORESIST COMPRISING PHOTOINITIATOR TO SURFACE OF SUBSTRATE; IMAGEWISE EXPOSING TO ACTINIC RADIATION TO PRODUCE EXPOSED AND NON-EXPOSED AREAS IN PHOTORESIST; TREATING WITH SAMPLE OF ALKALINE SOLUTION E. I. DU PONT DE NEMOURS AND COMPANY 2001-01-30 US claimed
EP-0941866-B1 Thermally imageable element having improved room light stability DU PONT (US) 2003-04-16 EP disclosed
EP-0909990-B1 Photopolymerizable compositions having improved sidewall geometry and development latitude DU PONT (US) 2002-10-16 EP disclosed
US-6180319-B1 APPLYING AQUEOUS-DEVELOPABLE PHOTORESIST COMPRISING PHOTOINITIATOR TO SURFACE OF SUBSTRATE; IMAGEWISE EXPOSING TO ACTINIC RADIATION TO PRODUCE EXPOSED AND NON-EXPOSED AREAS IN PHOTORESIST; TREATING WITH SAMPLE OF ALKALINE SOLUTION E. I. DU PONT DE NEMOURS AND COMPANY 2001-01-30 US disclosed
US-5962190-A BINDER OF C4-10 ALKYL METHACRYLATE, C4-10 ALKYL ACRYLATE, METHYL METHACRYLATE OR ETHYL METHACRYLATE, METHACRYLIC ACID OR ACRYLIC ACID, AND STYRENE; UNSATURATED CROSSLINKING AGENT; PHOTOINITIATOR; RELIEF IMAGES E. I. DU PONT DE NEMOURS AND COMPANY (US) 1999-10-05 US disclosed
EP-0941866-A1 Non-photosensitive, thermally imageable element having improved room light stability E. I. du Pont de Nemours and Company (US) 1999-09-15 EP disclosed
EP-0909990-A2 Photopolymerizable compositions having improved sidewall geometry and development latitude E.I. DU PONT DE NEMOURS AND COMPANY (US) 1999-04-21 EP disclosed