SCHEMBL7045274

SCHEMBL7045274

N=C(N)NCCC[C@H](C(=O)NCC(=O)O)N(Cc1ccc(CNC(N)=O)cc1)C(=O)Nc1cccc2ccccc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.42
GSK3B P49841 1/20 0.42
MC4R P32245 1/20 0.39
MC5R P33032 1/20 0.39
MC3R P41968 1/20 0.39
MC1R Q01726 1/20 0.39
ALDH1A1 P00352 2/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
GAA P10253 1/20 0.38
POLB P06746 1/20 0.37
TRPV1 Q8NER1 2/20 0.36
METAP2 P50579 1/20 0.36
METAP1 P53582 1/20 0.36
EPHX1 P07099 1/20 0.35
HSD17B10 Q99714 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
MMP1 P03956 1/20 0.35
MMP2 P08253 1/20 0.35
MMP9 P14780 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8528194 0.82 F7 (0.40) KDM4EMC4RMC5RMC3RMC1R
SCHEMBL8527067 0.82 ALDH1A1 (0.41) ALDH1A1MEN1KMT2AL3MBTL1
SCHEMBL8126001 0.79 F7 (0.44) KDM4EALDH1A1
SCHEMBL7040970 0.78 MMP1 (0.41) KDM4EGSK3BMC4RMC5RMC3R
SCHEMBL8526123 0.78 KMT2A (0.41) MC4RMC5RMC3RALDH1A1MEN1
SCHEMBL8526200 0.78 HDAC1 (0.35) POLB
SCHEMBL8526199 0.77 MC4R (0.40) MC4RMC5RMC3RMC1R
SCHEMBL7038757 0.76 NPY1R (0.38) MEN1KMT2A
SCHEMBL8526111 0.76 TMEM97 (0.38) ITGB3
SCHEMBL8528634 0.76 NPY1R (0.37) MEN1KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0885186-B1 AMINO ACID DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS AND PROCESSES FOR PREPARING THEM THOMAE GMBH DR K (DE) 2003-03-26 EP disclosed