SCHEMBL7045753

SCHEMBL7045753

COCCn1c(N2CCCNCC2)nc2c(OC(N)=O)cccc21

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 3/20 0.38
HTR2C P28335 2/20 0.37
ALDH1A1 P00352 3/20 0.37
CYP1A2 P05177 3/20 0.37
CASP1 P29466 3/20 0.37
HPGD P15428 2/20 0.37
CASP7 P55210 2/20 0.37
HSD17B10 Q99714 2/20 0.37
CHRNB2 P17787 1/20 0.36
CHRNA4 P43681 1/20 0.36
CYP3A4 P08684 2/20 0.36
HIF1A Q16665 2/20 0.36
CYP2C9 P11712 1/20 0.36
MEN1 O00255 1/20 0.36
USP2 O75604 1/20 0.36
KMT2A Q03164 1/20 0.36
PIK3CD O00329 1/20 0.36
SOS1 Q07889 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7041296 0.96 HTR3A (0.40) HTR3AHTR2CALDH1A1CYP1A2CASP1
SCHEMBL7044695 0.90 HTR3A (0.40) HTR3AHTR2CCHRNB2CHRNA4SOS1
SCHEMBL7036855 0.90 HTR3A (0.40) HTR3AHTR2CCHRNB2CHRNA4SOS1
SCHEMBL7042010 0.89 FLT3 (0.41) HTR3ACYP1A2CHRNB2CHRNA4CYP3A4
SCHEMBL7046777 0.88 HTR3A (0.39) HTR3ACHRNB2CHRNA4
SCHEMBL7037841 0.87 HTR3A (0.38) HTR3AHPGDMEN1KMT2A
SCHEMBL5621625 0.87 PARP1 (0.41) HTR3AHTR2C
SCHEMBL7043340 0.86 CHRNB2 (0.39) HTR3ACHRNB2CHRNA4MEN1KMT2A
SCHEMBL7042935 0.85 HTR3A (0.42) HTR3AHTR2CSOS1
SCHEMBL7042964 0.85 HTR3A (0.42) HTR3AHTR2CSOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133477-B1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS ABBOTT GMBH & CO KG (DE) 2004-02-18 EP disclosed