SCHEMBL7046986

SCHEMBL7046986

NC(=O)c1cccc2ncc(-c3ccc4ccccc4c3)nc12

nearest known ligand 0.70

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 17/20 0.70
PARP2 Q9UGN5 1/20 0.66
NOS1 P29475 1/20 0.47
CDC7 O00311 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7111338 0.85 PARP1 (0.80) PARP1PARP2
SCHEMBL7045348 0.84 PARP1 (0.69) PARP1PARP2
SCHEMBL7112515 0.83 PARP1 (1.00) PARP1PARP2
SCHEMBL7113559 0.82 PARP1 (0.67) PARP1PARP2CDC7
SCHEMBL424209 0.82 PARP1 (0.81) PARP1PARP2
SCHEMBL7045309 0.82 PARP1 (0.78) PARP1PARP2NOS1
SCHEMBL7042977 0.82 PARP1 (0.78) PARP1PARP2
SCHEMBL31602072 0.82 PARP1 (0.81) PARP1PARP2
SCHEMBL7115056 0.81 PARP1 (0.78) PARP1PARP2CDC7
SCHEMBL7045177 0.81 PARP1 (1.00) PARP1PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003007959-A1 QUINOXALINE DERIVATIVES WHICH HAVE PARP INHIBITORY ACTION FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-01-30 WO disclosed