SCHEMBL7049481

SCHEMBL7049481

CCS(=O)(=O)Nc1cc(N=C=O)c(F)cc1Br

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PSIP1 O75475 1/20 0.42
PGR P06401 4/20 0.34
HPGD P15428 2/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
LMNA P02545 1/20 0.33
HSD17B10 Q99714 1/20 0.33
BRAF P15056 3/20 0.32
AR P10275 1/20 0.31
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
MAPT P10636 1/20 0.30
JAK2 O60674 1/20 0.30
JAK1 P23458 1/20 0.30
TYK2 P29597 1/20 0.30
JAK3 P52333 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6662068 0.75 PSIP1 (0.47) PSIP1PGRHPGDCYP3A4CYP2C9
SCHEMBL31047810 0.72 PSIP1 (0.51) PSIP1PGRHPGDCYP3A4CYP2C9
SCHEMBL6199133 0.72 KMT2A (0.34)
SCHEMBL10519626 0.71 PSIP1 (0.41) PSIP1PGRHPGDLMNAHSD17B10
SCHEMBL5846557 0.71 CYP3A4 (0.42) HPGDCYP3A4ALDH1A1
SCHEMBL7688191 0.69 PGR (0.40) PSIP1PGRHPGDLMNAHSD17B10
SCHEMBL7017288 0.69 NEU3 (0.35) PGRARMAPT
SCHEMBL6663333 0.68 PSIP1 (0.50) PSIP1PGRHPGDLMNAHSD17B10
SCHEMBL30017045 0.67 CYP3A4 (0.42) HPGDCYP3A4ALDH1A1
SCHEMBL10938599 0.67 PPOX (0.32) CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030017948-A1 Method for producing n-substituted 2,4-diamino-5-fluoro benzonitriles and novel intermediates BAYER AKTIENGESELLSCHAFT (DE) 2003-01-23 US disclosed
EP-1244615-A1 METHOD FOR PRODUCING N-SUBSTITUTED 2,4-DIAMINO-5-FLUORO BENZONITRILES AND NOVEL INTERMEDIATES Bayer Aktiengesellschaft (DE) 2002-10-02 EP disclosed
WO-2001047873-A1 METHOD FOR PRODUCING N-SUBSTITUTED 2,4-DIAMINO-5-FLUORO BENZONITRILES AND NOVEL INTERMEDIATES BAYER AKTIENGESELLSCHAFT (DE) 2001-07-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030017948-A1 Method for producing n-substituted 2,4-diamino-5-fluoro benzonitriles and novel intermediates DDT, PFAS, DAO PSIP1 1439/4885PGR 4770/4885HPGD 1435/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.