SCHEMBL7053763

SCHEMBL7053763

CC(C)OC(OC(=O)CC(=O)O)OC(=O)CC(=O)O

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.33
LDHA P00338 1/20 0.33
SRR Q9GZT4 1/20 0.33
CYP1A2 P05177 1/20 0.32
LMNA P02545 2/20 0.31
MMP1 P03956 1/20 0.31
MMP2 P08253 1/20 0.31
MMP3 P08254 1/20 0.31
MMP9 P14780 1/20 0.31
MMP13 P45452 1/20 0.31
HCAR2 Q8TDS4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL242500 0.81 TSHR (0.47) TSHRLDHASRRLMNAMMP1
Benzene SCHEMBL28101101 0.77 TSHR (0.53) TSHRLDHASRRLMNAHCAR2
SCHEMBL8195362 0.77 TSHR (0.38) TSHRLDHASRRCYP1A2
SCHEMBL6270772 0.77 TSHR (0.38) TSHRLDHASRRCYP1A2
SCHEMBL28184861 0.77 MGAM (0.44) TSHRLMNA
Cyclopropane SCHEMBL29205269 0.76 TSHR (0.42) TSHRLDHASRRLMNAHCAR2
Alcohol SCHEMBL28450885 0.76 LMNA (0.45) TSHRLDHASRRLMNAHCAR2
Butane SCHEMBL452862 0.76 LMNA (0.50) TSHRLDHASRRLMNAHCAR2
SCHEMBL5349565 0.75 LDHA (0.38) TSHRLDHASRRCYP1A2LMNA
SCHEMBL1543387 0.74 THRB (0.42) TSHRLDHASRR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6653295-B2 Protease inhibitor; viricide BRISTOL-MYERS SQUIBB COMPANY 2003-11-25 US disclosed
US-20030064962-A1 Inhibitors of hepatitis C virus NS3 protease BRISTOL-MYERS SQUIBB COMPANY (FORMERLY D/B/A DUPONT PHARMACEUTICALS COMPANY) 2003-04-03 US disclosed
WO-2002048116-A2 INHIBITORS OF HEPATITIS C VIRUS NS3 PROTEASE BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2002-06-20 WO disclosed
EP-1037905-A1 ANTIPICORNAVIRAL COMPOUNDS AND METHODS FOR THEIR USE AND PREPARATION AGOURON PHARMACEUTICALS, INC. (US) 2000-09-27 EP disclosed
US-5962487-A PICORNAVIRAL 3C PROTEASE INHIBITORS AGOURON PHARMACEUTICALS, INC. (US) 1999-10-05 US disclosed
WO-1999031122-A9 ANTIPICORNAVIRAL COMPOUNDS AND METHODS FOR THEIR USE AND PREPARATION AGOURON PHARMA (US) 1999-09-30 WO disclosed
WO-1999031122-A1 ANTIPICORNAVIRAL COMPOUNDS AND METHODS FOR THEIR USE AND PREPARATION AGOURON PHARMACEUTICALS, INC. (US) 1999-06-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030064962-A1 Inhibitors of hepatitis C virus NS3 protease PRSS1, SERPINB1, SPINT2 TSHR 4782/4885LDHA 3285/4885SRR 392/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.