SCHEMBL7057796

SCHEMBL7057796

O=C(NCCCCN1CCC(Nc2cccc(C(F)(F)F)c2)CC1)c1cc2ccccc2[nH]1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 13/20 0.71
DRD2 P14416 11/20 0.71
HTR2A P28223 4/20 0.71
HTR1A P08908 3/20 0.71
HTR2C P28335 3/20 0.71
SLC6A2 P23975 1/20 0.57
SLC6A4 P31645 1/20 0.57
DRD4 P21917 4/20 0.54
KDM4E B2RXH2 2/20 0.52
HSD17B10 Q99714 2/20 0.52
AKR1C3 P42330 1/20 0.50
ALDH1A1 P00352 1/20 0.50
PLD2 O14939 1/20 0.49
HDAC3 O15379 1/20 0.49
HDAC4 P56524 1/20 0.49
HDAC1 Q13547 1/20 0.49
HDAC7 Q8WUI4 1/20 0.49
HDAC2 Q92769 1/20 0.49
HDAC10 Q969S8 1/20 0.49
HDAC11 Q96DB2 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7119593 0.84 CCR3 (0.55) DRD3DRD2ADRA1A
SCHEMBL7057584 0.84 DRD3 (0.69) DRD3DRD2SLC6A2SLC6A4DRD4
Hydrochloric Acid SCHEMBL7056135 0.83 DRD4 (0.59) DRD3DRD2HTR2AHTR1AHTR2C
SCHEMBL4525593 0.83 DRD2 (1.00) DRD3DRD2HTR2AHTR1AHTR2C
Hydrochloric Acid SCHEMBL7058141 0.81 DRD2 (0.53) DRD3DRD2HTR2AHTR1AHTR2C
SCHEMBL7053098 0.80 RAB9A (0.53) DRD3DRD2HTR2AHTR1AHTR2C
SCHEMBL7054406 0.80 DRD3 (0.57) DRD3DRD2HTR2AHTR1AHTR2C
SCHEMBL7055659 0.80 DRD2 (0.50) DRD3DRD2ADRA1A
SCHEMBL7060979 0.80 DRD2 (0.52) DRD3DRD2DRD4ADRA1A
SCHEMBL7052435 0.78 DRD2 (0.48) DRD3DRD2HTR2AHTR1AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003028725-A1 4-(1-PIPERIDINY)-BUTYLCARBOXAMIDE AS D3 DOPAMINE RECEPTOR SUBTYPE SELECTIVE LIGANDS Richter Gedeon Vegyészeti Gyár Rt. (HU) 2003-04-10 WO disclosed