SCHEMBL7066853

SCHEMBL7066853

CS(=O)(=O)Nc1cccc(Cl)c1Sc1ccc(Cl)cc1Cl

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 5/20 0.53
PTGS1 P23219 4/20 0.53
CCR2 P41597 5/20 0.45
NR3C1 P04150 3/20 0.43
NR3C2 P08235 3/20 0.43
PGR P06401 2/20 0.43
AR P10275 2/20 0.43
ITGB2 P05107 2/20 0.40
ICAM1 P05362 2/20 0.40
ITGAL P20701 2/20 0.40
KEAP1 Q14145 1/20 0.39
NFE2L2 Q16236 1/20 0.39
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.39
KMT2A Q03164 1/20 0.39
CYP2C9 P11712 1/20 0.38
AKR1B1 P15121 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7063649 0.79 PTGS1 (0.48) PTGS2PTGS1CCR2ITGB2ICAM1
SCHEMBL6598563 0.75 PTGS1 (0.58) PTGS2PTGS1CCR2ITGB2ICAM1
SCHEMBL4575696 0.73 PTGS1 (0.56) PTGS2PTGS1CCR2ITGB2ICAM1
SCHEMBL14906059 0.72 MCL1 (0.61) PTGS2PTGS1CCR2MAPT
SCHEMBL9538398 0.72 PTGS1 (0.55) PTGS2PTGS1CCR2ITGB2ICAM1
SCHEMBL8100630 0.71 CA2 (0.44) PTGS2PTGS1
SCHEMBL7979738 0.71 PTGS2 (0.56) PTGS2PTGS1CCR2ITGB2ICAM1
SCHEMBL9539406 0.71 PTGS1 (0.54) PTGS2PTGS1CCR2ITGB2ICAM1
SCHEMBL8481379 0.71 PTGS1 (0.43) PTGS2PTGS1CCR2ITGB2ICAM1
SCHEMBL11560825 0.71 MCL1 (0.59) PTGS2PTGS1CCR2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0968180-B1 SUBSTITUTED DERIVATIVES OF BENZOSULPHONAMIDES AS INHIBITORS OF THE ENZYME CYCLOOXYGENASE II NYCOMED AUSTRIA GMBH (AT) 2003-06-04 EP disclosed
US-6297282-B1 TREATING INFLAMMATION AND PAIN NYCOMED AUSTRIA GMBH (AT) 2001-10-02 US disclosed