SCHEMBL7068112

SCHEMBL7068112

CC(C[C@H](CC(=O)N[C@@H](Cc1ccccc1)C(=S)NCCCc1ccccc1)C(=O)O)c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 6/20 0.47
ACE P12821 1/20 0.44
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
KMT2A Q03164 2/20 0.43
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
MMP2 P08253 2/20 0.42
MMP7 P09237 2/20 0.42
MMP9 P14780 1/20 0.42
MMP12 P39900 1/20 0.42
MMP13 P45452 1/20 0.42
CNR1 P21554 1/20 0.42
POLB P06746 1/20 0.42
CTSG P08311 1/20 0.42
CMA1 P23946 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7068109 1.00 EPHX2 (0.47) EPHX2ACENPC1RAB9ASMN1; SMN2
SCHEMBL7982892 0.91 ACE (0.52) ACEKMT2AALDH1A1HPGDCYP2D6
SCHEMBL7982890 0.91 ACE (0.52) ACEKMT2AALDH1A1HPGDCYP2D6
SCHEMBL7068135 0.86 MMP2 (0.51) EPHX2MMP2MMP1MMP3
SCHEMBL7068140 0.86 MMP2 (0.51) EPHX2MMP2MMP1MMP3
SCHEMBL7135106 0.86 ACE (0.49) ACEMMP2MMP7MMP9MMP12
SCHEMBL27522992 0.86 MMP1 (0.49) HPGDMMP2MMP7MMP9CTSG
SCHEMBL7982632 0.86 MMP1 (0.49) HPGDMMP2MMP7MMP9CTSG
SCHEMBL27550386 0.85 MMP1 (0.46) EPHX2KMT2AALDH1A1HPGDCYP2D6
SCHEMBL7982631 0.84 EPHX2 (0.48) EPHX2ACEKMT2AALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1060161-B1 MATRIX METALLOPROTEINASE INHIBITORS LEO PHARMA AS WITH SECONDARY N (DK) 2003-06-11 EP disclosed
EP-1060161-A1 MATRIX METALLOPROTEINASE INHIBITORS LEO PHARMACEUTICAL PRODUCTS LTD. A/S (LOVENS KEMISKE FABRIK PRODUKTIONSAKTIESELSKAB) (DK) 2000-12-20 EP disclosed
WO-1999044989-A1 MATRIX METALLOPROTEINASE INHIBITORS LEO PHARMACEUTICAL PRODUCTS LTD. A/S (DK) 1999-09-10 WO disclosed