SCHEMBL7072308

SCHEMBL7072308

Nc1nc2nc(-c3cncs3)nc-2c[nH]1

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
IMPDH2 P12268 1/20 0.40
LATS1 O95835 1/20 0.32
CHEK1 O14757 1/20 0.32
CHEK2 O96017 1/20 0.32
PRMT5 O14744 1/20 0.32
WDR77 Q9BQA1 1/20 0.32
MYC P01106 1/20 0.31
IDO1 P14902 1/20 0.31
AR P10275 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6942143 0.68 CYP2A6 (0.37)
SCHEMBL7077154 0.67 HTR6 (0.41) PRMT5WDR77IDO1
SCHEMBL7075974 0.67 CCR1 (0.47)
SCHEMBL14320606 0.64 APP (0.50) IMPDH2CHEK1CHEK2PRMT5WDR77
SCHEMBL7070801 0.64 ADORA2A (0.44)
SCHEMBL8009682 0.63 METAP2 (0.44)
SCHEMBL6129041 0.62 NPC1 (0.46) IMPDH2CHEK1CHEK2MYC
SCHEMBL13822164 0.62 ASIC3 (0.47) IMPDH2MYCIDO1
SCHEMBL7071995 0.61 KDM4E (0.37)
SCHEMBL571374 0.61 HDAC8 (0.50) IMPDH2CHEK1CHEK2PRMT5WDR77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1349857-A1 PURINE DERIVATIVES AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2003-10-08 EP disclosed
WO-2002055521-A1 PURINE DERIVATIVES AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2002-07-18 WO disclosed