SCHEMBL7072708

SCHEMBL7072708

COc1ccc2c(Cc3ccc(Cl)c(Cl)c3)c(C(=O)O)[nH]c2c1

nearest known ligand 0.61

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GPR17 Q13304 3/20 0.61
BCL2 P10415 2/20 0.49
MCL1 Q07820 2/20 0.49
KDM4E B2RXH2 5/20 0.49
ALDH1A1 P00352 3/20 0.49
HPGD P15428 3/20 0.49
HSD17B10 Q99714 3/20 0.49
KMT2A Q03164 2/20 0.47
MEN1 O00255 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
POLB P06746 1/20 0.46
MDM2 Q00987 1/20 0.46
GAA P10253 2/20 0.46
CCR2 P41597 2/20 0.45
USP2 O75604 1/20 0.44
MAPT P10636 1/20 0.44
ALOX15 P16050 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7842628 0.80 KDM4E (0.47) BCL2MCL1KDM4EALDH1A1HPGD
SCHEMBL7592453 0.76 GPR35 (0.43) GPR17CYP2C9CYP2C19GAANPSR1
SCHEMBL9186531 0.76 GPR17 (1.00) GPR17KDM4EALDH1A1HPGDHSD17B10
SCHEMBL3659426 0.75 KDM4E (0.60) GPR17KDM4EALDH1A1HPGDHSD17B10
SCHEMBL1144751 0.73 GPR17 (0.64) GPR17KDM4EALDH1A1HPGDHSD17B10
SCHEMBL7680945 0.72 PTPRC (0.44) GPR17ALDH1A1HPGDMAPT
SCHEMBL7682574 0.72 KDM4A (0.43) GPR17ALDH1A1KMT2AMEN1CCR2
SCHEMBL7076761 0.72 MCL1 (0.48) GPR17BCL2MCL1KDM4EKMT2A
SCHEMBL30779683 0.72 GPR17 (0.63) GPR17KDM4EALDH1A1HPGDHSD17B10
SCHEMBL7074236 0.70 POLB (0.47) POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1003504-B1 INDOLE DERIVATIVES AND THEIR USE AS MCP-1 ANTAGONISTS ASTRAZENECA AB (SE) 2003-07-02 EP disclosed