SCHEMBL7073986

SCHEMBL7073986

N=C(N)c1ccc(C(=O)N2CCN(S(=O)(=O)Cc3ccccc3)CC2)cc1

nearest known ligand 0.62

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.62
ALDH1A1 P00352 4/20 0.58
PKM P14618 1/20 0.58
TSHR P16473 4/20 0.57
LMNA P02545 4/20 0.57
RAB9A P51151 1/20 0.57
GAA P10253 1/20 0.55
CYP2C19 P33261 1/20 0.55
SMN1; SMN2 Q16637 3/20 0.53
RECQL P46063 1/20 0.53
HIF1A Q16665 1/20 0.52
HSD11B1 P28845 1/20 0.51
KMT2A Q03164 1/20 0.50
HPGD P15428 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Acetic Acid SCHEMBL27550449 0.96 MAPK1 (0.58) MAPK1ALDH1A1PKMTSHRLMNA
SCHEMBL7075147 0.87 RAB9A (0.60) MAPK1ALDH1A1PKMTSHRLMNA
SCHEMBL7074220 0.81 LMNA (0.71) MAPK1ALDH1A1LMNAGAAKMT2A
SCHEMBL7069901 0.79 KDM4E (0.72) MAPK1ALDH1A1PKMTSHRLMNA
SCHEMBL5735712 0.79 MAPK1 (0.57) MAPK1ALDH1A1PKMTSHRLMNA
Acetic Acid SCHEMBL28744327 0.78 LMNA (0.70) ALDH1A1LMNAGAASMN1; SMN2KMT2A
SCHEMBL7070294 0.77 GAA (0.56) MAPK1ALDH1A1TSHRLMNAGAA
SCHEMBL7069417 0.77 HPGD (0.68) MAPK1ALDH1A1TSHRLMNASMN1; SMN2
SCHEMBL7071445 0.77 F10 (0.62) MAPK1ALDH1A1TSHRLMNAGAA
Acetic Acid SCHEMBL27568113 0.76 GAA (0.56) MAPK1ALDH1A1TSHRLMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1025086-B1 BENZAMIDINE DERIVATIVES AS FACTOR XA INHIBITORS MERCK PATENT GMBH (DE) 2003-06-25 EP disclosed
US-6492368-B1 Benzamidine derivatives as factor XA inhibitors MERCK PATENT GMBH (DE) 2002-12-10 US disclosed