SCHEMBL7075147

SCHEMBL7075147

N=C(N)c1ccc(CC(=O)N2CCN(S(=O)(=O)Cc3ccccc3)CC2)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 1/20 0.60
ALDH1A1 P00352 4/20 0.56
TSHR P16473 2/20 0.56
LMNA P02545 2/20 0.56
SMN1; SMN2 Q16637 2/20 0.53
MAPK1 P28482 2/20 0.53
GAA P10253 2/20 0.52
CYP2C19 P33261 1/20 0.52
F2 P00734 2/20 0.52
PRSS1 P07477 2/20 0.52
TPSAB1 Q15661 1/20 0.52
TPSD1 Q9BZJ3 1/20 0.52
TPSG1 Q9NRR2 1/20 0.52
GLA P06280 1/20 0.52
PKM P14618 2/20 0.50
CNR1 P21554 1/20 0.49
KMT2A Q03164 2/20 0.49
F10 P00742 1/20 0.48
PRSS2 P07478 1/20 0.48
PRSS3 P35030 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7073986 0.87 MAPK1 (0.62) RAB9AALDH1A1TSHRLMNASMN1; SMN2
SCHEMBL7074851 0.85 GAA (0.63) ALDH1A1TSHRLMNAGAAF2
Acetic Acid SCHEMBL27550449 0.84 MAPK1 (0.58) RAB9AALDH1A1TSHRLMNASMN1; SMN2
SCHEMBL7074218 0.82 ALDH1A1 (0.67) ALDH1A1TSHRSMN1; SMN2MAPK1GAA
SCHEMBL7367810 0.80 RAB9A (0.48) RAB9AALDH1A1TSHRLMNASMN1; SMN2
SCHEMBL7654785 0.80 YAP1 (0.61) ALDH1A1TSHRLMNASMN1; SMN2GAA
SCHEMBL7076859 0.80 YAP1 (0.61) ALDH1A1TSHRLMNASMN1; SMN2GAA
SCHEMBL7075829 0.79 F2 (0.49) ALDH1A1TSHRLMNASMN1; SMN2GAA
SCHEMBL7074652 0.79 F2 (0.54) ALDH1A1TSHRSMN1; SMN2GAAF2
SCHEMBL7074867 0.78 TGM2 (0.55) ALDH1A1TSHRLMNAGAAF2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1025086-B1 BENZAMIDINE DERIVATIVES AS FACTOR XA INHIBITORS MERCK PATENT GMBH (DE) 2003-06-25 EP disclosed
US-6492368-B1 Benzamidine derivatives as factor XA inhibitors MERCK PATENT GMBH (DE) 2002-12-10 US disclosed