SCHEMBL7074159

SCHEMBL7074159

Cc1nc(-c2ccc(C(=O)N3CCN(C(=O)c4cccnc4)CC3)cc2)no1

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 1/20 0.55
MAPK1 P28482 1/20 0.53
TDP1 Q9NUW8 1/20 0.51
ABL1 P00519 3/20 0.50
BCR P11274 3/20 0.50
PKM P14618 1/20 0.50
FABP6 P51161 1/20 0.50
HDAC4 P56524 1/20 0.50
HDAC2 Q92769 1/20 0.50
HDAC8 Q9BY41 1/20 0.50
HDAC6 Q9UBN7 1/20 0.50
MYC P01106 1/20 0.50
POLB P06746 1/20 0.49
MKNK1 Q9BUB5 1/20 0.49
MKNK2 Q9HBH9 1/20 0.49
MEN1 O00255 1/20 0.48
MAPT P10636 1/20 0.48
KMT2A Q03164 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7074772 0.84 MGLL (0.66) MGLLMAPK1HDAC4HDAC2HDAC8
SCHEMBL7384950 0.80 FABP6 (0.46) MGLLMAPK1FABP6
SCHEMBL7076687 0.80 TSHR (0.59) MGLLHDAC4HDAC2HDAC8HDAC6
SCHEMBL13838154 0.80 ALDH1A1 (0.53) MGLLMAPK1ABL1BCRPKM
SCHEMBL7071414 0.79 FASN (0.60) MGLLHDAC4HDAC2HDAC8HDAC6
SCHEMBL7075196 0.79 MGLL (0.54) MGLLMAPK1HDAC4HDAC2HDAC8
SCHEMBL9763711 0.78 PKM (0.74) MAPK1TDP1PKMFABP6POLB
SCHEMBL7074230 0.78 HPGD (0.53) MGLLPKMHDAC4HDAC2HDAC8
SCHEMBL7071696 0.77 ALDH1A1 (0.61) MGLLHDAC4HDAC2HDAC8HDAC6
SCHEMBL7649408 0.77 DGAT1 (0.58) MGLLHDAC4POLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1025086-B1 BENZAMIDINE DERIVATIVES AS FACTOR XA INHIBITORS MERCK PATENT GMBH (DE) 2003-06-25 EP disclosed
US-6492368-B1 Benzamidine derivatives as factor XA inhibitors MERCK PATENT GMBH (DE) 2002-12-10 US disclosed