SCHEMBL7076508

SCHEMBL7076508

COc1ccc(CNS(=O)(=O)Cc2ccccc2C(=O)NO)cc1

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.52
MMP13 P45452 9/20 0.52
MMP9 P14780 7/20 0.52
MMP8 P22894 5/20 0.52
MMP12 P39900 5/20 0.52
MMP2 P08253 4/20 0.52
MMP14 P50281 4/20 0.52
MMP16 P51512 4/20 0.52
MMP1 P03956 6/20 0.49
MMP3 P08254 3/20 0.49
SLC6A5 Q9Y345 1/20 0.47
HPGD P15428 3/20 0.47
ALDH1A1 P00352 2/20 0.47
OPRK1 P41145 1/20 0.47
ADAM17 P78536 2/20 0.46
TSHR P16473 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7076482 0.89 HTT (0.56) HTTHPGDALDH1A1OPRK1TSHR
SCHEMBL7072870 0.88 HTT (0.58) HTTSLC6A5HPGDALDH1A1OPRK1
SCHEMBL7072113 0.81 MMP2 (0.63) HTTMMP13MMP9MMP8MMP12
SCHEMBL5898955 0.81 MMP9 (0.62) MMP13MMP9MMP8MMP12MMP2
SCHEMBL7076512 0.77 MMP9 (0.53) MMP13MMP9MMP8MMP12MMP2
SCHEMBL8413524 0.75 HTT (0.65) HTTALDH1A1OPRK1TSHR
SCHEMBL25839479 0.74 HPGD (0.68) HTTSLC6A5HPGDALDH1A1
SCHEMBL7076489 0.73 MMP12 (0.68) HTTMMP13MMP9MMP8MMP12
SCHEMBL22230464 0.72 HTT (0.65) HTTALDH1A1TSHR
SCHEMBL27811168 0.71 TSHR (0.73) HTTHPGDALDH1A1OPRK1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030022893-A1 Hydroxamic and carboxylic acid derivatives BAXTER ANDREW DOUGLAS (GB) 2003-01-30 US claimed
US-6465468-B1 SUCH AS N-HYDROXY-2-(4-(4-CHLOROPHENYL)PIPERAZINE-1-SULFONYL)BENZAMIDE; INHIBITORS OF MATRIX METALLOPROTEINASE, ADAM OR ADAMTS ENZYMES; TREATMENT OF DEGENERATIVE DISEASES AND CERTAIN CANCERS DARWIN DISCOVERY LIMITED (GB) 2002-10-15 US claimed
US-20030022893-A1 Hydroxamic and carboxylic acid derivatives BAXTER ANDREW DOUGLAS (GB) 2003-01-30 US disclosed
US-6465468-B1 SUCH AS N-HYDROXY-2-(4-(4-CHLOROPHENYL)PIPERAZINE-1-SULFONYL)BENZAMIDE; INHIBITORS OF MATRIX METALLOPROTEINASE, ADAM OR ADAMTS ENZYMES; TREATMENT OF DEGENERATIVE DISEASES AND CERTAIN CANCERS DARWIN DISCOVERY LIMITED (GB) 2002-10-15 US disclosed