SCHEMBL7076535

SCHEMBL7076535

O=C(O)Oc1c(Cl)c2cc(F)ccc2n1Cc1ccc(Cl)c(Cl)c1

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 15/20 0.56
ABCB11 O95342 4/20 0.51
TBXA2R P21731 1/20 0.46
KDM4E B2RXH2 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
MAPT P10636 1/20 0.43
CYP2C9 P11712 1/20 0.43
HPGD P15428 1/20 0.43
TSHR P16473 1/20 0.43
CYP2C19 P33261 1/20 0.43
HIF1A Q16665 1/20 0.43
HSD17B10 Q99714 1/20 0.43
PTGES2 Q9H7Z7 1/20 0.43
TDP1 Q9NUW8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6307041 0.82 CCR2 (0.72) CCR2ABCB11TBXA2R
SCHEMBL7077464 0.77 CCR2 (0.53) CCR2ABCB11TBXA2R
SCHEMBL6300631 0.77 CCR2 (0.52) CCR2ABCB11TBXA2RKDM4ECYP1A2
SCHEMBL7072402 0.76 CCR2 (0.59) CCR2ABCB11CYP1A2CYP3A4MAPT
SCHEMBL7076337 0.76 CCR2 (0.69) CCR2ABCB11TBXA2R
SCHEMBL11466147 0.74 CCR2 (0.55) CCR2ABCB11TBXA2RKDM4ECYP1A2
SCHEMBL9239098 0.74 ALDH1A1 (0.42) KDM4EHPGDHSD17B10
SCHEMBL9238617 0.73 MEN1 (0.41) CCR2CYP1A2CYP3A4MAPTCYP2C9
SCHEMBL7080358 0.73 CCR2 (0.70) CCR2ABCB11CYP1A2CYP3A4MAPT
SCHEMBL11459984 0.73 CCR2 (0.50) CCR2ABCB11TBXA2RKDM4ECYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1003504-B1 INDOLE DERIVATIVES AND THEIR USE AS MCP-1 ANTAGONISTS ASTRAZENECA AB (SE) 2003-07-02 EP claimed