SCHEMBL7078045

SCHEMBL7078045

O=C1c2cccc3cccc(c23)N1c1ccc[nH]1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE6D O43924 1/20 0.52
KMT2A Q03164 4/20 0.49
MEN1 O00255 3/20 0.49
ALDH1A1 P00352 4/20 0.46
HPGD P15428 3/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
CASP1 P29466 2/20 0.46
MPI P34949 1/20 0.46
CACNA1B Q00975 1/20 0.46
APBA1 Q02410 1/20 0.46
KDM4E B2RXH2 4/20 0.43
POLB P06746 1/20 0.42
ERCC1 P07992 1/20 0.42
FEN1 P39748 1/20 0.42
ERCC4 Q92889 1/20 0.42
GAA P10253 3/20 0.42
CASP7 P55210 1/20 0.41
LMNA P02545 2/20 0.40
HTT P42858 2/20 0.40
L3MBTL1 Q9Y468 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28358758 0.89 ALDH1A1 (0.50) KMT2AMEN1ALDH1A1HPGDSMN1; SMN2
SCHEMBL10869116 0.76 PDE6D (0.81) PDE6DKMT2AMEN1ALDH1A1HPGD
SCHEMBL2865639 0.76 KMT2A (0.42) KMT2AMEN1ALDH1A1POLBHTT
SCHEMBL28190986 0.76 CES1 (0.56) ALDH1A1GAA
SCHEMBL9290287 0.73 PDE6D (0.82) PDE6DKMT2AMEN1ALDH1A1HPGD
SCHEMBL30267 0.73 CES1 (0.38) KMT2AMEN1ALDH1A1POLBGAA
SCHEMBL1101925 0.71 KMT2A (0.62) PDE6DKMT2AMEN1ALDH1A1HPGD
SCHEMBL9290288 0.70 ALDH1A1 (0.79) PDE6DKMT2AMEN1ALDH1A1HPGD
SCHEMBL9290285 0.70 PDE6D (0.61) PDE6DKMT2AMEN1ALDH1A1HPGD
SCHEMBL24317276 0.70 PDE6D (0.50) PDE6DKMT2AMEN1ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1358180-A2 NAPHTHOSTYRIL DERIVATIVES AND THEIR USE AS INHIBITORS OF CYCLIN-DEPENDENT KINASES F. Hoffmann-La Roche AG (CH) 2003-11-05 EP disclosed
WO-2002059109-A2 NAPHTHOSTYRIL DERIVATIVES AND THEIR USE AS INHIBITORS OF CYCLIN- DEPENDENT KINASES F. HOFFMANN-LA ROCHE AG (CH) 2002-08-01 WO disclosed