SCHEMBL30267

SCHEMBL30267

C=C1C(=O)N(c2ccc[nH]2)c2ccccc21

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CES1 P23141 5/20 0.38
ALDH1A1 P00352 2/20 0.38
BCHE P06276 2/20 0.38
CES2 O00748 1/20 0.38
GAA P10253 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
MGLL Q99685 1/20 0.34
NR1H3 Q13133 7/20 0.34
NR1H2 P55055 6/20 0.34
POLB P06746 1/20 0.33
TTR P02766 1/20 0.33
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
ATM Q13315 1/20 0.32
TGM2 P21980 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14334422 0.77 HIF1A (0.39) CES1ALDH1A1BCHECES2GAA
SCHEMBL2865639 0.77 KMT2A (0.42) ALDH1A1NR1H3NR1H2POLBMEN1
SCHEMBL8443315 0.74 ALDH1A1 (0.67) CES1ALDH1A1BCHECES2GAA
SCHEMBL25433322 0.74 HIPK2 (0.44) CES1ALDH1A1BCHECES2GAA
SCHEMBL7078045 0.73 PDE6D (0.52) ALDH1A1GAAPOLBMEN1KMT2A
SCHEMBL8098957 0.73 KDR (0.39) CES1ALDH1A1BCHECES2GAA
SCHEMBL1990739 0.72 TDP2 (0.31)
SCHEMBL16862997 0.67 POLB (0.50) CES1ALDH1A1NR1H3NR1H2POLB
SCHEMBL28358758 0.67 ALDH1A1 (0.50) CES1ALDH1A1BCHECES2GAA
SCHEMBL31107472 0.66 TTR (0.64) CES1ALDH1A1NR1H3NR1H2TTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1641435-A2 RATE CONTROLLED RELEASE OF A PHARMACEUTICAL AGENT IN A BIODEGRADABLE DEVICE BAUSCH & LOMB INCORPORATED (US) 2006-04-05 EP claimed
US-20050031669-A1 Rate controlled release of a pharmaceutical agent in a biodegradable device BAUSCH & LOMB INCORPORATED (US) 2005-02-10 US claimed
WO-2004112748-A2 RATE CONTROLLED RELEASE OF A PHARMACEUTICAL AGENT IN A BIODEGRADABLE DEVICE BAUSCH & LOMB INCORPORATED (US) 2004-12-29 WO claimed
US-20040253293-A1 Rate controlled release of a pharmaceutical agent in a biodegradable device BAUSCH & LOMB INCORPORATED 2004-12-16 US claimed
WO-2012025726-A1 Novel Hybrid Compounds UNIVERSITY OF GREENWICH (GB) 2012-03-01 WO disclosed
EP-1641435-A2 RATE CONTROLLED RELEASE OF A PHARMACEUTICAL AGENT IN A BIODEGRADABLE DEVICE BAUSCH & LOMB INCORPORATED (US) 2006-04-05 EP disclosed
US-20050031669-A1 Rate controlled release of a pharmaceutical agent in a biodegradable device BAUSCH & LOMB INCORPORATED (US) 2005-02-10 US disclosed
WO-2004112748-A2 RATE CONTROLLED RELEASE OF A PHARMACEUTICAL AGENT IN A BIODEGRADABLE DEVICE BAUSCH & LOMB INCORPORATED (US) 2004-12-29 WO disclosed
US-20040253293-A1 Rate controlled release of a pharmaceutical agent in a biodegradable device BAUSCH & LOMB INCORPORATED 2004-12-16 US disclosed