SCHEMBL7078874

SCHEMBL7078874

CN(C)c1cc(CCN)cc(C(F)(F)F)c1

nearest known ligand 0.50

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 2/20 0.50
MAOB P27338 4/20 0.42
NOS1 P29475 3/20 0.40
NOS2 P35228 3/20 0.40
IDO1 P14902 2/20 0.38
TACR1 P25103 4/20 0.37
HTR2A P28223 2/20 0.37
NOS3 P29474 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7074326 0.86 IDO1 (0.40) TAAR1MAOBNOS1NOS2IDO1
SCHEMBL626371 0.81 TAAR1 (0.64) TAAR1MAOBIDO1HTR2A
SCHEMBL14117328 0.80 SIGMAR1 (0.40) NOS1NOS2IDO1TACR1
Hydrochloric Acid SCHEMBL1970957 0.79 TAAR1 (0.62) TAAR1MAOBIDO1HTR2A
SCHEMBL3950720 0.79 MRGPRX4 (0.38) NOS1NOS2IDO1TACR1
SCHEMBL3950360 0.79 RXRA (0.42) IDO1TACR1
SCHEMBL7694014 0.77 TACR1 (0.43) IDO1TACR1
SCHEMBL16515444 0.77 TAAR1 (0.55) TAAR1MAOBNOS1NOS2IDO1
SCHEMBL806196 0.74 TAAR1 (0.56) TAAR1MAOBIDO1HTR2A
SCHEMBL43792 0.74 TAAR1 (0.56) TAAR1MAOBIDO1HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030036653-A1 Diaminopyridine-containing thiourea inhibitors of herpes viruses AMERICAN HOME PRODUCTS CORPORATION 2003-02-20 US disclosed
US-20020026055-A1 Aminopyridine-containing thiourea inhibitors of herpes viruses AMERICAN HOME PRODUCTS CORPORATION 2002-02-28 US disclosed
US-20010039348-A1 Alpha-methylbenzyl-containing thiourea inhibitors of herpes viruses containing a phenylenediamine group AMERICAN HOME PRODUCTS CORPORATION (US) 2001-11-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030036653-A1 Diaminopyridine-containing thiourea inhibitors of herpes viruses HAVCR2, CCR6, CXCR6 TAAR1 211/4885MAOB 3776/4885NOS1 4151/4885
US-20010039348-A1 Alpha-methylbenzyl-containing thiourea inhibitors of herpes viruses containing a phenylenediamine group CCR6, HAVCR2, BCOR TAAR1 407/4885MAOB 2576/4885NOS1 2473/4885
US-20020026055-A1 Aminopyridine-containing thiourea inhibitors of herpes viruses TK1, TPMT, CXCR6 TAAR1 1159/4885MAOB 4517/4885NOS1 3126/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.