SCHEMBL7080474

SCHEMBL7080474

CC(C)c1[nH]c(C(Cc2ccncc2)OCCO)nc1Sc1cccc(Cl)c1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSNK2A2 P19784 1/20 0.34
CSNK2B P67870 1/20 0.34
ADRB2 P07550 1/20 0.33
ADRB1 P08588 1/20 0.33
ADRB3 P13945 1/20 0.33
ALDH1A1 P00352 3/20 0.32
KMT2A Q03164 2/20 0.32
KDM4E B2RXH2 2/20 0.32
HPGD P15428 2/20 0.32
MEN1 O00255 1/20 0.32
MAPT P10636 2/20 0.32
POLB P06746 1/20 0.32
PPP1CA P62136 1/20 0.32
ALOX12 P18054 1/20 0.31
PDE4D Q08499 1/20 0.31
PDE4B Q07343 1/20 0.31
LMNA P02545 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6974065 0.92
SCHEMBL7086505 0.89 MAPK13 (0.30)
SCHEMBL6972450 0.89 CDK5 (0.32) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL6960607 0.87 ALOX12 (0.36) ALDH1A1KMT2AKDM4EHPGDMEN1
SCHEMBL6957342 0.86 CSNK2A2 (0.38) CSNK2A2CSNK2BALDH1A1KMT2AKDM4E
SCHEMBL7084598 0.86 ADRB2 (0.33) CSNK2A2CSNK2BADRB2ADRB1ADRB3
SCHEMBL6961323 0.85 PDE4B (0.35) ALDH1A1KMT2AHPGDMEN1MAPT
SCHEMBL7082933 0.85 CSNK2A2 (0.38) CSNK2A2CSNK2BALDH1A1KMT2AKDM4E
SCHEMBL6967186 0.84
SCHEMBL6964726 0.84 ALDH1A1 (0.36) ADRB2ADRB1ADRB3ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed