SCHEMBL7082933

SCHEMBL7082933

CC(C)c1[nH]c(C(O)Cc2ccncc2)nc1Sc1cccc(Cl)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSNK2A2 P19784 1/20 0.38
CSNK2B P67870 1/20 0.38
ALDH1A1 P00352 4/20 0.36
HPGD P15428 3/20 0.36
KMT2A Q03164 3/20 0.36
KDM4E B2RXH2 2/20 0.36
MEN1 O00255 2/20 0.36
POLB P06746 2/20 0.35
LMNA P02545 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
SLC2A1 P11166 2/20 0.34
MAPT P10636 3/20 0.33
PPP1CA P62136 1/20 0.33
FNTA P49354 1/20 0.33
FNTB P49356 1/20 0.33
PDE5A O76074 1/20 0.33
PDE9A O76083 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6968179 0.90 CYP1A2 (0.33) CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL6974320 0.88 MAPK14 (0.34) CYP3A4SMN1; SMN2TP53TYMS
SCHEMBL6973409 0.87 SLC6A4 (0.36) ALDH1A1KMT2ACYP1A2CYP3A4CYP2C9
SCHEMBL7087098 0.86 TP53 (0.39) ALDH1A1HPGDKMT2AKDM4EMEN1
SCHEMBL6957342 0.86 CSNK2A2 (0.38) CSNK2A2CSNK2BALDH1A1HPGDKMT2A
SCHEMBL7080474 0.85 CSNK2A2 (0.34) CSNK2A2CSNK2BALDH1A1HPGDKMT2A
SCHEMBL7079911 0.83 SLC2A1 (0.34) CSNK2A2CSNK2BALDH1A1HPGDKMT2A
SCHEMBL6968078 0.83 ALOX5 (0.38) ALDH1A1HPGDKMT2AMEN1LMNA
SCHEMBL6972114 0.83 LMNA (0.41) CSNK2A2CSNK2BALDH1A1HPGDKMT2A
SCHEMBL6973795 0.83 GSK3B (0.32) KMT2AMEN1POLBCYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed