SCHEMBL7081241

SCHEMBL7081241

CC(=O)NCc1nc(C(C)C)c(Sc2cccc(F)c2)n1Cc1ccncc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.36
LMNA P02545 2/20 0.36
ENPP2 Q13822 4/20 0.35
S1PR3 Q99500 1/20 0.35
MAPT P10636 2/20 0.35
GRIN1 Q05586 1/20 0.35
GRIN2B Q13224 1/20 0.35
ALDH1A1 P00352 1/20 0.35
POLB P06746 1/20 0.35
RECQL P46063 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HSD17B10 Q99714 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
ADORA3 P0DMS8 1/20 0.35
ADORA2A P29274 1/20 0.35
ADORA2B P29275 1/20 0.35
ADORA1 P30542 1/20 0.35
ROCK2 O75116 1/20 0.35
ROCK1 Q13464 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7087801 0.92 ROCK2 (0.36) TP53LMNAENPP2S1PR3MAPT
SCHEMBL7082084 0.92 ENPP2 (0.35) TP53LMNAENPP2S1PR3MAPT
SCHEMBL7086202 0.90 LMNA (0.41) LMNAENPP2S1PR3GRIN1GRIN2B
SCHEMBL6974067 0.90 POLB (0.38) TP53LMNAMAPTALDH1A1POLB
SCHEMBL7086493 0.89 GRIN1 (0.35) TP53LMNAENPP2S1PR3GRIN1
SCHEMBL7082255 0.89 ALDH1A1 (0.41) TP53S1PR3MAPTALDH1A1POLB
SCHEMBL7084176 0.87 SMN1; SMN2 (0.38) ALDH1A1POLBSMN1; SMN2L3MBTL1
SCHEMBL8109545 0.87 GRIN1 (0.36) TP53LMNAGRIN1GRIN2BALDH1A1
SCHEMBL6967611 0.86 GRIN1 (0.35) TP53LMNAS1PR3MAPTGRIN1
SCHEMBL6973952 0.86 ENPP2 (0.36) TP53LMNAENPP2MAPTGRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed