SCHEMBL7081563

SCHEMBL7081563

COc1ccc2c3c(sc2c1)-c1ccccc1C3

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.45
CA2 P00918 2/20 0.45
CA4 P22748 2/20 0.45
CA6 P23280 2/20 0.45
ALDH1A1 P00352 2/20 0.42
CYP3A4 P08684 2/20 0.42
MAPT P10636 2/20 0.42
CYP2C19 P33261 2/20 0.42
HSD17B10 Q99714 2/20 0.42
TSHR P16473 2/20 0.42
MAPK1 P28482 2/20 0.42
KDM4E B2RXH2 1/20 0.42
TP53 P04637 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
PKM P14618 1/20 0.42
HPGD P15428 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
ACHE P22303 2/20 0.41
DRD2 P14416 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7074787 0.77 LIMK1 (0.44) CA1CA2CA4CA6ACHE
SCHEMBL7077021 0.70 HSP90AA1 (0.45) ALDH1A1CYP3A4MAPTCYP2C19HSD17B10
SCHEMBL7107233 0.69 HSP90AA1 (0.53) ALDH1A1CYP3A4MAPTCYP2C19HSD17B10
SCHEMBL29771277 0.69 ESR1 (0.43) ALDH1A1CYP3A4MAPTCYP2C19HSD17B10
SCHEMBL2294178 0.69 CA1 (0.73) CA1CA2CA4CA6ALDH1A1
SCHEMBL7102544 0.69 MAPT (0.53) ALDH1A1CYP3A4MAPTCYP2C19HSD17B10
SCHEMBL27261519 0.69 ESR1 (0.43) ALDH1A1CYP3A4MAPTCYP2C19HSD17B10
SCHEMBL2914928 0.69 DRD1 (0.58) CA1CA2CA4CA6ALDH1A1
SCHEMBL3287680 0.69 ALDH1A1 (0.56) CA1CA2CA4CA6ALDH1A1
SCHEMBL29633762 0.69 DRD1 (0.58) CA1CA2CA4CA6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832891-B1 Dihydrobenzo (B) indeno (2,1-D) thiophene compounds, intermediates, processes, compositions, and methods LILLY CO ELI (US) 2003-07-30 EP disclosed
EP-0832891-A1 Dihydrobenzo (B) indeno (2,1-D) thiophene compounds, intermediates, processes, compositions, and methods ELI LILLY AND COMPANY (US) 1998-04-01 EP disclosed