SCHEMBL6974232

SCHEMBL6974232

CC(C)c1nc(CCN)n(Cc2ccncc2)c1Sc1cccc(Cl)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.35
TDP1 Q9NUW8 3/20 0.34
TAAR1 Q96RJ0 1/20 0.33
ALDH1A1 P00352 3/20 0.33
KDM4E B2RXH2 2/20 0.33
HPGD P15428 2/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.32
KCNH2 Q12809 1/20 0.32
POLB P06746 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
PDE4D Q08499 1/20 0.32
GSK3B P49841 1/20 0.32
NPC1 O15118 1/20 0.32
PDE4B Q07343 1/20 0.32
TLR7 Q9NYK1 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6967360 0.92 IDO1 (0.36) IDO1TDP1ALDH1A1KDM4EHPGD
SCHEMBL7082703 0.91 KCNH2 (0.34) TDP1KCNH2GSK3BTLR7PIM1
SCHEMBL6971118 0.91 ALDH1A1 (0.37) TDP1TAAR1ALDH1A1KDM4EHPGD
SCHEMBL6959029 0.90 IDO1 (0.35) IDO1TDP1ALDH1A1KDM4ELMNA
SCHEMBL6975055 0.89 GRIN1 (0.35) TAAR1LMNAKMT2AL3MBTL1GSK3B
SCHEMBL7082836 0.89 TLR7 (0.38) TDP1ALDH1A1KDM4EMAPTGSK3B
SCHEMBL7083480 0.88 TLR8 (0.37) IDO1TDP1ALDH1A1KDM4EHPGD
SCHEMBL7079909 0.88 IDO1 (0.36) IDO1TDP1ALDH1A1KDM4EHPGD
SCHEMBL6967782 0.87 LMNA (0.39) IDO1TDP1ALDH1A1KDM4ELMNA
SCHEMBL7084720 0.86 HTR3E (0.40) IDO1TDP1TAAR1ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed