SCHEMBL7082902

SCHEMBL7082902

C#CCC(=O)c1ccc(F)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.57
RAB9A P51151 2/20 0.57
PTPN1 P18031 1/20 0.57
HTR7 P34969 1/20 0.50
CES2 O00748 1/20 0.50
CES1 P23141 1/20 0.50
PLOD2 O00469 1/20 0.50
HSD11B1 P28845 2/20 0.49
CA1 P00915 2/20 0.46
CA2 P00918 2/20 0.46
MEN1 O00255 1/20 0.44
MAPT P10636 1/20 0.44
HPGD P15428 1/20 0.44
ALOX12 P18054 1/20 0.44
HTT P42858 1/20 0.44
KMT2A Q03164 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
BCL2L1 Q07817 1/20 0.43
BAD Q92934 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fluorobenzene SCHEMBL28684421 0.86 HSD11B1 (0.49) NPC1RAB9APTPN1CES1HSD11B1
SCHEMBL133680 0.81 NPC1 (0.55) NPC1RAB9APTPN1HTR7CES2
SCHEMBL28581878 0.78 GSK3B (0.59) NPC1RAB9ACES2CES1HSD11B1
Benzene SCHEMBL28690163 0.77 MAPK1 (0.58) NPC1RAB9APTPN1CES2CES1
SCHEMBL7085528 0.77 MAPK1 (0.58) NPC1RAB9APTPN1CES2CES1
SCHEMBL2491432 0.77 PLOD2 (0.69) NPC1RAB9APTPN1HTR7CES2
SCHEMBL26584242 0.77 NPC1 (0.82) NPC1RAB9APTPN1HTR7CES2
SCHEMBL11571 0.75 NPC1 (0.64) NPC1RAB9APTPN1HTR7CES2
SCHEMBL1094528 0.75 NPC1 (0.64) NPC1RAB9APTPN1HTR7CES2
SCHEMBL1266504 0.75 NPC1 (0.64) NPC1RAB9APTPN1HTR7CES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1051413-B1 QUINOLINE DERIVATIVES AS ANTIBACTERIALS SMITHKLINE BEECHAM PLC (GB) 2003-06-04 EP claimed
EP-0548664-B1 2,3,3a-5,9b-hexahydro-1H-benzo(e)indole derivatives HOFFMANN LA ROCHE (CH) 1995-05-31 EP claimed
EP-0232089-B1 QUINONE AMIDES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1991-03-13 EP claimed
EP-0100046-B1 CIS-4A-ARYL-1,2,3,4,4A,9B-HEXAHYDRO-BENZOFURO(3,2-C)PYRIDINES, A PROCESS FOR PREPARING THE SAME, AND THEIR USE AS MEDICAMENTS HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1988-02-03 EP claimed
EP-0002283-B1 SUBSTITUTED 1,3-DIHYDROSPIRO (BENZO(C)THIOPHENES), PROCESS FOR THEIR PREPARATION AND THESE COMPOUNDS FOR USE AS MEDICAMENTS HOECHST AKTIENGESELLSCHAFT (DE) 1983-08-24 EP claimed