SCHEMBL7085263

SCHEMBL7085263

COc1cccc(CN2CCN(c3cc4ccccc4n3S(=O)(=O)c3ccccc3)CC2)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.56
LMNA P02545 5/20 0.54
HTT P42858 1/20 0.54
HTR6 P50406 2/20 0.54
TSHR P16473 3/20 0.51
HTR1A P08908 1/20 0.51
DRD2 P14416 1/20 0.51
HTR2B P41595 1/20 0.51
ALOX15 P16050 1/20 0.51
ALDH1A1 P00352 5/20 0.49
KDM4E B2RXH2 3/20 0.49
GAA P10253 2/20 0.49
CASP1 P29466 1/20 0.48
CASP4 P49662 1/20 0.48
CASP5 P51878 1/20 0.48
MAPK1 P28482 1/20 0.47
FAAH O00519 1/20 0.47
MAPT P10636 2/20 0.46
MEN1 O00255 1/20 0.46
RECQL P46063 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7085731 0.88 HTR6 (0.53) SIGMAR1LMNAHTR6TSHRHTR1A
SCHEMBL1537840 0.77 HTR6 (0.78) HTR6HTR1ADRD2
SCHEMBL7086820 0.74 HTR6 (0.55) HTR6DRD2
SCHEMBL8570664 0.73 SIGMAR1 (0.81) SIGMAR1LMNATSHRDRD2ALDH1A1
SCHEMBL20804357 0.73 SIGMAR1 (0.90) SIGMAR1LMNAHTTTSHRHTR1A
SCHEMBL28186295 0.73 SIGMAR1 (0.90) SIGMAR1LMNAHTTTSHRHTR1A
SCHEMBL4304442 0.71 HTR6 (0.54) HTR6HTR1ADRD2
SCHEMBL8174066 0.71 SIGMAR1 (0.71) SIGMAR1LMNATSHRHTR1ADRD2
Hydrochloric Acid SCHEMBL4316251 0.70 HTR6 (0.53) HTR6HTR1ADRD2
Hydrochloric Acid SCHEMBL6521806 0.70 HTR6 (0.53) HTR6HTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1343756-A2 1-ARYL- OR 1-ALKYLSULFONYL-HETEROCYCLYLBENZAZOLES AS 5-HYDROXYTRYPTAMINE-6 LIGANDS Wyeth (US) 2003-09-17 EP disclosed
WO-2002036562-A2 1-ARYL- OR 1-ALKYLSULFONYL-HETEROCYCLYLBENZAZOLES AS 5-HYDROXYTRYPTAMINE-6 LIGANDS WYETH (US) 2002-05-10 WO disclosed