SCHEMBL7086820

SCHEMBL7086820

O=S(=O)(c1ccccc1Br)n1c(N2CCN(Cc3ccccc3)CC2)cc2ccccc21

nearest known ligand 0.55

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 12/20 0.55
CHRM1 P11229 1/20 0.50
DRD2 P14416 1/20 0.46
DRD4 P21917 1/20 0.43
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
TRPV4 Q9HBA0 1/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA9 Q16790 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7085731 0.85 HTR6 (0.53) HTR6DRD2DRD4CYP2D6
SCHEMBL6829699 0.76 HTR6 (0.60) HTR6CHRM1CYP3A4CYP2D6
SCHEMBL7085263 0.74 SIGMAR1 (0.56) HTR6DRD2
SCHEMBL1537822 0.72 HTR6 (0.75) HTR6CHRM1CYP3A4CYP2D6
SCHEMBL3561901 0.70 ACLY (0.46) HTR6CHRM1CA12CA1CA2
SCHEMBL3563939 0.70 ACLY (0.62) CA12CA2CA9
SCHEMBL3223044 0.67 HTR6 (1.00) HTR6CHRM1CYP3A4CYP2D6
SCHEMBL3409661 0.67 HTR6 (1.00) HTR6CHRM1CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL3219058 0.66 HTR6 (0.98) HTR6CHRM1CYP3A4CYP2D6
SCHEMBL4304442 0.65 HTR6 (0.54) HTR6DRD2CYP3A4CA12CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1343756-A2 1-ARYL- OR 1-ALKYLSULFONYL-HETEROCYCLYLBENZAZOLES AS 5-HYDROXYTRYPTAMINE-6 LIGANDS Wyeth (US) 2003-09-17 EP disclosed
WO-2002036562-A2 1-ARYL- OR 1-ALKYLSULFONYL-HETEROCYCLYLBENZAZOLES AS 5-HYDROXYTRYPTAMINE-6 LIGANDS WYETH (US) 2002-05-10 WO disclosed