SCHEMBL7085318

SCHEMBL7085318

CC(C)c1nc(C=NO)n(Cc2ccccn2)c1Sc1ccccc1

nearest known ligand 0.34

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.34
ALOX5AP P20292 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
GABRA1 P14867 1/20 0.32
GABRA5 P31644 1/20 0.32
TP53 P04637 3/20 0.31
KDM4E B2RXH2 3/20 0.31
ALOX15 P16050 1/20 0.31
HTT P42858 1/20 0.31
HSD17B10 Q99714 1/20 0.31
CYP1A2 P05177 1/20 0.30
CYP2C19 P33261 1/20 0.30
S1PR3 Q99500 2/20 0.30
NPC1 O15118 1/20 0.30
LMNA P02545 1/20 0.30
RAB9A P51151 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
HRH1 P35367 1/20 0.30
TLR7 Q9NYK1 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7085317 1.00 ALDH1A1 (0.34) ALDH1A1ALOX5APPTGDR2GABRA1GABRA5
SCHEMBL6969251 0.90 GRIN1 (0.38) ALDH1A1S1PR3RAB9ASMN1; SMN2
SCHEMBL6971733 0.90 GRM5 (0.35) ALDH1A1TP53KDM4EHTTCYP1A2
SCHEMBL6969252 0.90 GRIN1 (0.38) ALDH1A1S1PR3RAB9ASMN1; SMN2
SCHEMBL6971738 0.90 GRM5 (0.35) ALDH1A1TP53KDM4EHTTCYP1A2
SCHEMBL7084152 0.89 S1PR3 (0.34) ALDH1A1ALOX5APKDM4ES1PR3LMNA
SCHEMBL6969160 0.89 ADRA1D (0.32) ALDH1A1ALOX5APTP53KDM4ES1PR3
SCHEMBL6969157 0.89 ADRA1D (0.32) ALDH1A1ALOX5APTP53KDM4ES1PR3
SCHEMBL7084149 0.89 S1PR3 (0.34) ALDH1A1ALOX5APKDM4ES1PR3LMNA
SCHEMBL6973368 0.86 ALDH1A1 (0.34) ALDH1A1ALOX5APPTGDR2GABRA1GABRA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed