SCHEMBL7085754

SCHEMBL7085754

CCCc1c[nH]c2ccc(Oc3c(C(F)(F)F)cc(N)cc3C(F)(F)F)cc12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRA P10827 5/20 0.48
THRB P10828 5/20 0.48
HTR1A P08908 10/20 0.48
HTR1B P28222 10/20 0.48
HTR1D P28221 9/20 0.46
TRPM8 Q7Z2W7 2/20 0.46
HTR2A P28223 3/20 0.46
MAPT P10636 3/20 0.46
CYP1A2 P05177 2/20 0.46
TSHR P16473 1/20 0.46
NFKB1 P19838 1/20 0.46
HTR2C P28335 1/20 0.46
HTR7 P34969 1/20 0.46
HTR6 P50406 1/20 0.46
HTR4 Q13639 1/20 0.46
MAPK1 P28482 2/20 0.46
TDP1 Q9NUW8 2/20 0.46
KDM4E B2RXH2 1/20 0.46
TP53 P04637 1/20 0.46
CYP3A4 P08684 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7085031 0.93 HTR1A (0.50) THRATHRBHTR1AHTR1BHTR1D
SCHEMBL7087277 0.92 HTR1B (0.52) THRATHRBHTR1AHTR1BHTR1D
SCHEMBL7088178 0.91 THRA (0.52) THRATHRBHTR1AHTR1BHTR1D
SCHEMBL7088760 0.85 THRA (0.52) THRATHRBHTR1AHTR1BHTR1D
SCHEMBL7088959 0.84 LTA4H (0.48) THRATHRBHTR1AHTR1BHTR1D
SCHEMBL7089278 0.83 HTR1A (0.52) THRATHRBHTR1AHTR1BHTR1D
SCHEMBL7090401 0.83 HTR1A (0.52) HTR1AHTR1BHTR1DTRPM8HTR2A
SCHEMBL6860169 0.83 THRA (0.71) THRATHRBHTR1AHTR1BHTR1D
SCHEMBL7089913 0.83 THRA (0.47) THRATHRBHTR1AHTR1BHTR1D
SCHEMBL7089914 0.83 THRA (0.47) THRATHRBHTR1AHTR1BHTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1268422-A1 INDOLES FOR TREATING DISEASES THAT CAN BE TREATED USING THYROID HORMONES Bayer Aktiengesellschaft (DE) 2003-01-02 EP disclosed
WO-2001070687-A1 INDOLES FOR TREATING DISEASES THAT CAN BE TREATED USING THYROID HORMONES BAYER AKTIENGESELLSCHAFT (DE) 2001-09-27 WO disclosed