SCHEMBL7090401

SCHEMBL7090401

CCCc1c[nH]c2ccc(Oc3c(Br)cc(N)cc3Br)cc12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 10/20 0.52
HTR1B P28222 9/20 0.52
HTR1D P28221 8/20 0.50
HTR2A P28223 3/20 0.50
MAPT P10636 3/20 0.50
TRPM8 Q7Z2W7 2/20 0.50
CYP1A2 P05177 2/20 0.50
TSHR P16473 1/20 0.50
NFKB1 P19838 1/20 0.50
HTR2C P28335 1/20 0.50
HTR7 P34969 1/20 0.50
HTR6 P50406 1/20 0.50
HTR4 Q13639 1/20 0.50
MAPK1 P28482 2/20 0.49
TDP1 Q9NUW8 2/20 0.49
CYP2D6 P10635 2/20 0.49
KDM4E B2RXH2 1/20 0.49
TP53 P04637 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2C9 P11712 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7090377 0.93 HTR1A (0.54) HTR1AHTR1BHTR1DHTR2AMAPT
SCHEMBL7084332 0.92 HTR1B (0.56) HTR1AHTR1BHTR1DHTR2AMAPT
SCHEMBL7088686 0.91 HTR1B (0.57) HTR1AHTR1BHTR1DHTR2AMAPT
SCHEMBL7089278 0.88 HTR1A (0.52) HTR1AHTR1BHTR1DHTR2AMAPT
SCHEMBL7084434 0.84 LTA4H (0.50) HTR1AHTR1BHTR1DHTR2AMAPT
SCHEMBL7085754 0.83 THRA (0.48) HTR1AHTR1BHTR1DHTR2AMAPT
SCHEMBL6862010 0.83 KDM4E (0.53) HTR1AHTR1BHTR1DKDM4EMEN1
SCHEMBL6985214 0.82 CYP2D6 (0.45) HTR1AHTR1BHTR1DHTR2AMAPT
SCHEMBL6515562 0.82 MTNR1A (0.50) HTR1AHTR1BHTR1DHTR2ACYP1A2
SCHEMBL7088630 0.80 THRA (0.47) HTR1AHTR1BHTR1DHTR2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1268422-A1 INDOLES FOR TREATING DISEASES THAT CAN BE TREATED USING THYROID HORMONES Bayer Aktiengesellschaft (DE) 2003-01-02 EP disclosed
WO-2001070687-A1 INDOLES FOR TREATING DISEASES THAT CAN BE TREATED USING THYROID HORMONES BAYER AKTIENGESELLSCHAFT (DE) 2001-09-27 WO disclosed