SCHEMBL7086840

SCHEMBL7086840

O=C(Cc1ccncn1)Nc1ccc(NC(=O)c2ccccc2-c2ccccc2C(F)(F)F)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.44
PTPRC P08575 1/20 0.43
CHRNB2 P17787 1/20 0.43
CHRNB4 P30926 1/20 0.43
CHRNA3 P32297 1/20 0.43
CHRNA4 P43681 1/20 0.43
F2R P25116 1/20 0.42
SGMS2 Q8NHU3 1/20 0.42
KDR P35968 2/20 0.41
AURKA O14965 1/20 0.41
AURKB Q96GD4 1/20 0.41
RORC P51449 2/20 0.40
TRPV1 Q8NER1 1/20 0.40
TYK2 P29597 1/20 0.40
ATR Q13535 1/20 0.40
HTT P42858 1/20 0.40
MPL P40238 1/20 0.40
ANO1 Q5XXA6 1/20 0.40
CYP3A4 P08684 2/20 0.40
CYP2C9 P11712 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6791612 0.87 ALDH1A1 (0.52) ALDH1A1CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL7086836 0.84 TYK2 (0.47) ALDH1A1CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL7086824 0.79 LMNA (0.48) ALDH1A1CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL27631122 0.77 EPHX2 (0.53) ALDH1A1HTTCYP2C9TSHRHSD17B10
SCHEMBL6792281 0.75 SMO (0.62) ALDH1A1KDRTRPV1HTTLMNA
SCHEMBL7086831 0.75 CHRNB2 (0.43) ALDH1A1CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL7085677 0.73 LMNA (0.45) PTPRCTRPV1LMNA
SCHEMBL7085416 0.72 ADRB3 (0.48) ALDH1A1SGMS2HTTCYP3A4LMNA
SCHEMBL1826907 0.70 S1PR1 (0.50) ALDH1A1PTPRCAURKAAURKBTRPV1
SCHEMBL6795383 0.69 LMNA (0.52) ALDH1A1TRPV1HTTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1326835-A1 BENZAMIDE COMPOUNDS AS APO B SECRETION INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-07-16 EP disclosed
WO-2002028835-A1 BENZAMIDE COMPOUNDS AS APO B SECRETION INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-04-11 WO disclosed