SCHEMBL7086994

SCHEMBL7086994

COC(=O)[C@H](CC(C)(C)C)NC(=O)OCc1ccc(C)nc1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CTSL P07711 3/20 0.47
CTSB P07858 3/20 0.47
CTSS P25774 1/20 0.47
KYNU Q16719 1/20 0.41
ALDH1A1 P00352 2/20 0.39
ALOX15 P16050 1/20 0.39
POLB P06746 1/20 0.39
ITGB3 P05106 2/20 0.38
ITGA2B P08514 2/20 0.38
CYP3A4 P08684 1/20 0.36
TSHR P16473 1/20 0.36
MBOAT4 Q96T53 1/20 0.36
ATM Q13315 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6983383 0.91 CTSL (0.50) CTSLCTSBCTSSITGB3ITGA2B
SCHEMBL3044553 0.80 CTSS (0.70) CTSLCTSBCTSSKYNUALDH1A1
SCHEMBL33526968 0.77 KLK5 (0.50) CTSLCTSBCTSSITGB3ITGA2B
SCHEMBL7384652 0.77 CTSK (0.52) CTSLCTSBCTSS
SCHEMBL12241473 0.77 KLK5 (0.50) CTSLCTSBCTSSITGB3ITGA2B
SCHEMBL7086316 0.75 NPC1 (0.52) CTSLCTSBCTSSKYNUALDH1A1
SCHEMBL8169761 0.74 ITGB3 (0.50) CTSLCTSBCTSSALDH1A1ALOX15
SCHEMBL7303468 0.74 TYR (0.46) CTSLCTSBCTSSPOLBTSHR
SCHEMBL7303476 0.74 TYR (0.46) CTSLCTSBCTSSPOLBTSHR
SCHEMBL25516818 0.74 CTSL (0.53) CTSLCTSBCTSSKYNUALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1093367-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2003-03-05 EP disclosed
EP-1093367-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2001-04-25 EP disclosed
WO-1999066925-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1999-12-29 WO disclosed