SCHEMBL7087005

SCHEMBL7087005

N#Cc1cccc(NC2(OC(=O)O)CCSCC2)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.45
MAPT P10636 3/20 0.45
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
CYP2D6 P10635 3/20 0.44
HSD17B10 Q99714 3/20 0.44
HIF1A Q16665 2/20 0.43
GAA P10253 1/20 0.43
ALOX15 P16050 1/20 0.43
CASP7 P55210 1/20 0.43
CYP3A4 P08684 6/20 0.42
CYP1A2 P05177 4/20 0.42
CYP2C9 P11712 4/20 0.42
CYP2C19 P33261 4/20 0.42
USP2 O75604 4/20 0.42
TSHR P16473 3/20 0.42
HTT P42858 1/20 0.41
LMNA P02545 1/20 0.41
MAPK1 P28482 5/20 0.41
GRM5 P41594 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7087140 0.85 ALDH1A1 (0.42) ALDH1A1MAPTMEN1KMT2ACYP2D6
SCHEMBL7083930 0.81 ALDH1A1 (0.51) ALDH1A1MAPTMEN1KMT2ACYP2D6
SCHEMBL7089649 0.79 PGR (0.43) MAPTCYP2D6HIF1ACYP3A4CYP1A2
SCHEMBL7137822 0.76 CYP2D6 (0.41) ALDH1A1CYP2D6HSD17B10HIF1ACYP3A4
SCHEMBL6989644 0.71 ALDH1A1 (0.51) ALDH1A1MAPTMEN1KMT2ACYP2D6
SCHEMBL6991506 0.71 MAPT (0.50) MAPTGAAHTTLMNAMAPK1
SCHEMBL6991463 0.70 TSHR (0.51) ALDH1A1MAPTMEN1KMT2ACYP2D6
SCHEMBL7076644 0.68 HIF1A (0.48) ALDH1A1MAPTMEN1KMT2ACYP2D6
SCHEMBL7081753 0.68 LMNA (0.52) ALDH1A1MAPTMEN1KMT2ACYP2D6
SCHEMBL30606801 0.67 MAPT (0.87) ALDH1A1MAPTMEN1KMT2AHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1303482-A2 N-SUBSTITUTED-1-AMINO-1,1-DIALKYLCARBOXYLIC ACID DERIVATIVES MERCK PATENT GmbH (DE) 2003-04-23 EP disclosed
WO-2002008177-A2 N-SUBSTITUTED-1-AMINO-1,1-DIALKYLCARBOXYLIC ACID DERIVATIVES MERCK PATENT GMBH (DE) 2002-01-31 WO disclosed