SCHEMBL7089649

SCHEMBL7089649

N#Cc1cccc(S(=O)(=O)NC2(OC(=O)O)CCSCC2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PGR P06401 1/20 0.43
KAT6A Q92794 3/20 0.42
DPP4 P27487 1/20 0.40
DPP7 Q9UHL4 1/20 0.40
ACLY P53396 2/20 0.40
BRD4 O60885 1/20 0.39
RXFP1 Q9HBX9 1/20 0.38
CCKBR P32239 1/20 0.38
USP2 O75604 2/20 0.38
CYP1A2 P05177 2/20 0.38
CYP3A4 P08684 2/20 0.38
HIF1A Q16665 1/20 0.38
ITGAV P06756 1/20 0.37
GLO1 Q04760 1/20 0.37
SLC40A1 Q9NP59 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
TSHR P16473 1/20 0.37
MAPK1 P28482 1/20 0.37
CYP2C19 P33261 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7090243 0.87 MMP1 (0.44) PGRKAT6AACLYCCKBRITGAV
SCHEMBL7084134 0.83 KAT6A (0.44) PGRKAT6ADPP4DPP7ACLY
SCHEMBL7087005 0.79 ALDH1A1 (0.45) USP2CYP1A2CYP3A4HIF1ACYP2D6
SCHEMBL6994772 0.74 USP2 (0.53) PGRKAT6AACLYCCKBRUSP2
SCHEMBL6990928 0.73 USP2 (0.55) PGRKAT6AACLYCCKBRUSP2
SCHEMBL16108775 0.72 PARG (0.59) PGRKAT6AACLYBRD4RXFP1
SCHEMBL7077236 0.71 MMP1 (0.52) PGRKAT6AACLYUSP2CYP1A2
SCHEMBL30367627 0.71 PGR (0.46) PGRKAT6AACLYBRD4RXFP1
SCHEMBL7078089 0.70 USP2 (0.44) PGRKAT6AACLYCCKBRUSP2
SCHEMBL27589461 0.70 CYP3A4 (0.48) PGRKAT6ADPP4DPP7CCKBR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1303482-A2 N-SUBSTITUTED-1-AMINO-1,1-DIALKYLCARBOXYLIC ACID DERIVATIVES MERCK PATENT GmbH (DE) 2003-04-23 EP disclosed
WO-2002008177-A2 N-SUBSTITUTED-1-AMINO-1,1-DIALKYLCARBOXYLIC ACID DERIVATIVES MERCK PATENT GMBH (DE) 2002-01-31 WO disclosed