SCHEMBL7089116

SCHEMBL7089116

CC(C)[C@@H](CS(=O)(=O)N1CCN(c2ccc(-c3ccc(F)cc3)cn2)CC1)C(=O)N1C(=O)OCC1Cc1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.38
DRD4 P21917 1/20 0.38
HTR2A P28223 1/20 0.38
SLC6A4 P31645 1/20 0.38
DRD3 P35462 1/20 0.38
RORC P51449 2/20 0.35
IDH1 O75874 7/20 0.34
LMNA P02545 2/20 0.34
POLB P06746 1/20 0.34
NAMPT P43490 2/20 0.34
TNF P01375 1/20 0.34
STAT3 P40763 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
NOD2 Q9HC29 1/20 0.34
NOD1 Q9Y239 1/20 0.34
ADAMTS4 O75173 1/20 0.34
CYP3A4 P08684 1/20 0.34
MMP13 P45452 1/20 0.34
MMP14 P50281 1/20 0.34
KCNH2 Q12809 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6786463 1.00 HTR1A (0.38) HTR1ADRD4HTR2ASLC6A4DRD3
SCHEMBL6788834 1.00 HTR1A (0.38) HTR1ADRD4HTR2ASLC6A4DRD3
SCHEMBL6782817 0.93 RORC (0.35) RORCIDH1LMNANAMPTTNF
SCHEMBL7090855 0.93 RORC (0.35) RORCIDH1LMNANAMPTTNF
SCHEMBL6831648 0.93 RORC (0.35) RORCIDH1LMNANAMPTTNF
SCHEMBL6782024 0.92 LMNA (0.34) RORCIDH1LMNAPOLBNAMPT
SCHEMBL6782020 0.92 LMNA (0.34) RORCIDH1LMNAPOLBNAMPT
Hydrochloric Acid SCHEMBL7177099 0.88 CYP3A4 (0.33) IDH1LMNAPOLBNAMPTSMN1; SMN2
Hydrochloric Acid SCHEMBL7177094 0.88 CYP3A4 (0.33) IDH1LMNAPOLBNAMPTSMN1; SMN2
SCHEMBL6781731 0.86 TDO2 (0.40) IDH1NAMPTKCNH2PPARADGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1282614-A1 HYDROXAMIC ACID DERIVATIVES Darwin Discovery Limited (GB) 2003-02-12 EP disclosed
WO-2001087870-A1 HYDROXAMIC ACID DERIVATIVES DARWIN DISCOVERY LIMITED (GB) 2001-11-22 WO disclosed