SCHEMBL7092115

SCHEMBL7092115

COc1ccc(NC(C)=O)cc1C1OCCO1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.51
RORC P51449 1/20 0.46
NR3C1 P04150 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2C19 P33261 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
HPGD P15428 1/20 0.45
POLB P06746 1/20 0.45
HTT P42858 3/20 0.44
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
MAPK1 P28482 2/20 0.44
LMNA P02545 1/20 0.44
ALOX15 P16050 1/20 0.44
CHRNB2 P17787 1/20 0.44
CHRNA4 P43681 1/20 0.44
MAPT P10636 3/20 0.43
KDM4E B2RXH2 1/20 0.43
NPC1 O15118 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28252352 0.80 TDP1 (0.55) ALDH1A1RORCCYP1A2CYP2C19NPSR1
SCHEMBL7091504 0.78 NR3C1 (0.48) NR3C1CYP1A2RAB9A
SCHEMBL28518947 0.77 RORC (0.51) ALDH1A1RORCCYP1A2CYP2C19NPSR1
SCHEMBL1851780 0.75 SMN1; SMN2 (0.68) ALDH1A1CYP1A2CYP2C19POLBHTT
SCHEMBL30492996 0.75 SMN1; SMN2 (0.68) ALDH1A1CYP1A2CYP2C19POLBHTT
SCHEMBL7092393 0.74 NPC1 (0.42) ALDH1A1NPSR1POLBHTTMEN1
SCHEMBL829610 0.74 TGM2 (0.49) ALDH1A1MEN1KMT2ASMN1; SMN2LMNA
SCHEMBL28520661 0.73 CYP1A2 (0.43) ALDH1A1CYP1A2CYP2C19NPSR1POLB
SCHEMBL5952099 0.72 ALDH1A1 (0.62) ALDH1A1RORCPOLBHTTMEN1
SCHEMBL13414995 0.72 SMN1; SMN2 (0.52) ALDH1A1CYP1A2CYP2C19NPSR1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0665843-B1 SUBSTITUTED QUINUCLIDINES AS SUBSTANCE P ANTAGONISTS PFIZER (US) 2003-08-13 EP disclosed
US-5837711-A Substituted quinuclidines as substance P antagonists PFIZER INC. (US) 1998-11-17 US disclosed
EP-0665843-A1 SUBSTITUTED QUINUCLIDINES AS SUBSTANCE P ANTAGONISTS PFIZER INC. (US) 1995-08-09 EP disclosed
WO-1994010170-A1 SUBSTITUTED QUINUCLIDINES AS SUBSTANCE P ANTAGONISTS PFIZER INC. (US) 1994-05-11 WO disclosed