SCHEMBL7092393

SCHEMBL7092393

COc1ccc(N(C)C(C)=O)cc1C1OCCO1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.42
POLB P06746 2/20 0.42
AHR P35869 1/20 0.42
ALDH1A1 P00352 3/20 0.36
HTT P42858 1/20 0.36
ALOX5 P09917 1/20 0.36
RAB9A P51151 1/20 0.36
MTNR1A P48039 1/20 0.35
MTNR1B P49286 1/20 0.35
LMNA P02545 2/20 0.35
KDM4E B2RXH2 1/20 0.35
HSD17B10 Q99714 1/20 0.35
L3MBTL1 Q9Y468 2/20 0.34
MIF P14174 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
MAPT P10636 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
TDP1 Q9NUW8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7088720 0.78 NR3C1 (0.46) NPC1ALDH1A1RAB9ALMNAKDM4E
SCHEMBL7092115 0.74 ALDH1A1 (0.51) NPC1POLBALDH1A1HTTRAB9A
SCHEMBL29404113 0.74 MAPT (0.41) NPC1ALDH1A1HTTRAB9ALMNA
SCHEMBL9796263 0.73 POLB (0.49) NPC1POLBAHRALDH1A1HTT
SCHEMBL7093467 0.71 ACHE (0.48) NPC1POLBALDH1A1HTTRAB9A
SCHEMBL7090123 0.70 KDM4E (0.42) NPC1ALDH1A1HTTRAB9ALMNA
SCHEMBL19308888 0.70 MEN1 (0.51) NPC1POLBAHRALDH1A1HTT
SCHEMBL1670216 0.70 MEN1 (0.47) NPC1POLBALDH1A1HTTRAB9A
SCHEMBL13503862 0.70 ALDH1A1 (0.48) NPC1POLBAHRALDH1A1HTT
SCHEMBL7053663 0.70 NPC1 (0.39) NPC1ALDH1A1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0665843-B1 SUBSTITUTED QUINUCLIDINES AS SUBSTANCE P ANTAGONISTS PFIZER (US) 2003-08-13 EP disclosed
US-5837711-A Substituted quinuclidines as substance P antagonists PFIZER INC. (US) 1998-11-17 US disclosed
EP-0665843-A1 SUBSTITUTED QUINUCLIDINES AS SUBSTANCE P ANTAGONISTS PFIZER INC. (US) 1995-08-09 EP disclosed
WO-1994010170-A1 SUBSTITUTED QUINUCLIDINES AS SUBSTANCE P ANTAGONISTS PFIZER INC. (US) 1994-05-11 WO disclosed