SCHEMBL7092445

SCHEMBL7092445

COC(=O)C(Cc1cc(Br)c(OCCCCN=C(NC(=O)OC(C)(C)C)NC(=O)OC(C)(C)C)c(Br)c1)=NOCc1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPFFR1 Q9GZQ6 2/20 0.39
NPFFR2 Q9Y5X5 2/20 0.39
CA2 P00918 8/20 0.39
CA1 P00915 5/20 0.39
THRB P10828 7/20 0.38
THRA P10827 5/20 0.38
KLK7 P49862 1/20 0.35
KLK5 Q9Y337 1/20 0.35
NR1H4 Q96RI1 1/20 0.34
CA9 Q16790 2/20 0.33
CA12 O43570 1/20 0.33
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
BLM P54132 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7141370 0.79 NPFFR1 (0.40) NPFFR1NPFFR2CA2CA1KLK7
SCHEMBL7093257 0.77 MAPT (0.39) CA2CA1CA9CA12MEN1
SCHEMBL7093258 0.77 MAPT (0.39) CA2CA1CA9CA12MEN1
SCHEMBL7091866 0.77 CA1 (0.42) NPFFR1NPFFR2CA2CA1THRB
SCHEMBL7091722 0.73 CA2 (0.48) CA2CA1CA9CA12MEN1
SCHEMBL7091721 0.73 CA2 (0.48) CA2CA1CA9CA12MEN1
SCHEMBL7093259 0.71 LTA4H (0.43) CA2CA1CA9CA12KDM4E
SCHEMBL7089757 0.67 CA2 (0.44) CA2CA1CA9CA12
SCHEMBL7089756 0.67 CA2 (0.44) CA2CA1CA9CA12
SCHEMBL7093260 0.66 CA2 (0.35) CA2CA1CA9CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003087127-A2 ANTIMICROBIAL COMPOUNDS AGAINST STAPHYLOCOCCI, MYCOBACTERIA, AND OTHER INFECTIOUS AGENTS EXEGENICS INC. (US) 2003-10-23 WO disclosed