SCHEMBL7093259

SCHEMBL7093259

COC(=O)C(Cc1cc(Cl)c(OCCC(N)C(=O)OC(C)(C)C)c(Cl)c1)=NOCc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 3/20 0.43
CA2 P00918 7/20 0.35
CA1 P00915 4/20 0.35
LMNA P02545 1/20 0.35
CA9 Q16790 4/20 0.34
CA12 O43570 2/20 0.33
ITGA4 P13612 1/20 0.33
ITGB7 P26010 1/20 0.33
MAPT P10636 2/20 0.33
NPSR1 Q6W5P4 2/20 0.33
PSMB5 P28074 1/20 0.33
KDM4E B2RXH2 1/20 0.33
MAPK1 P28482 1/20 0.33
CTSL P07711 1/20 0.33
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7093257 0.83 MAPT (0.39) CA2CA1LMNACA9CA12
SCHEMBL7093258 0.83 MAPT (0.39) CA2CA1LMNACA9CA12
SCHEMBL7093260 0.81 CA2 (0.35) LTA4HCA2CA1LMNACA9
SCHEMBL7089757 0.75 CA2 (0.44) CA2CA1LMNACA9CA12
SCHEMBL7089756 0.75 CA2 (0.44) CA2CA1LMNACA9CA12
SCHEMBL7092445 0.71 NPFFR1 (0.39) CA2CA1CA9CA12MAPT
SCHEMBL29447511 0.69 LTA4H (0.57) LTA4HPSMB5
SCHEMBL7141370 0.68 NPFFR1 (0.40) CA2CA1CA9CA12MAPT
SCHEMBL7092580 0.67 CA2 (0.59) CA2CA1LMNACA9CA12
SCHEMBL7092581 0.67 CA2 (0.59) CA2CA1LMNACA9CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003087127-A2 ANTIMICROBIAL COMPOUNDS AGAINST STAPHYLOCOCCI, MYCOBACTERIA, AND OTHER INFECTIOUS AGENTS EXEGENICS INC. (US) 2003-10-23 WO disclosed